SCHEMBL904091

SCHEMBL904091

CCc1cnc(N2C[C@H]3C[C@H](Br)C[C@H]3C2)nc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 14/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
OGA O60502 1/20 0.35
PDE8B O95263 1/20 0.33
HDAC3 O15379 2/20 0.32
HDAC4 P56524 2/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC7 Q8WUI4 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC10 Q969S8 2/20 0.32
HDAC11 Q96DB2 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC9 Q9UKV0 2/20 0.32
HDAC5 Q9UQL6 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10068057 0.90 NPC1 (0.40) GPR119KDM4ENPC1RAB9AOGA
SCHEMBL904089 0.84 NPC1 (0.36) GPR119KDM4ENPC1RAB9AOGA
SCHEMBL10067572 0.80 ACACB (0.44) GPR119KDM4ENPC1RAB9AOGA
SCHEMBL10067707 0.80 ACACB (0.44) GPR119KDM4ENPC1RAB9AOGA
SCHEMBL18794991 0.76 HDAC3 (0.35) KDM4ENPC1RAB9AHDAC3HDAC4
SCHEMBL20064433 0.76 HRH3 (0.41) GPR119KDM4ENPC1RAB9AOGA
SCHEMBL12525218 0.76 OGA (0.38) GPR119KDM4ENPC1RAB9AOGA
SCHEMBL904079 0.76 KDM4E (0.42) GPR119KDM4ENPC1RAB9A
SCHEMBL23744766 0.73 PTPN11 (0.41) GPR119KDM4ENPC1RAB9AOGA
SCHEMBL10067598 0.73 HDAC3 (0.37) GPR119KDM4ENPC1RAB9AOGA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed