SCHEMBL9040971

SCHEMBL9040971

CC(N)C(=O)c1cccc(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.58
CHRNA1 P02708 1/20 0.56
CHRNG P07510 1/20 0.56
CHRNB1 P11230 1/20 0.56
CHRNB2 P17787 1/20 0.56
SLC6A2 P23975 1/20 0.56
CHRNB4 P30926 1/20 0.56
CHRNA3 P32297 1/20 0.56
CHRNA4 P43681 1/20 0.56
SLC6A3 Q01959 1/20 0.56
CHRND Q07001 1/20 0.56
ALDH1A1 P00352 3/20 0.50
SMN1; SMN2 Q16637 7/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
CASP3 P42574 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
C1S P09871 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL22557048 0.98 PARP1 (0.56) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL28007604 0.85 PARP1 (0.62) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL29922182 0.85 CHRNA1 (0.59) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL3125040 0.85 CHRNA1 (0.59) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL2599175 0.83 CHRNA1 (0.58) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL30310283 0.83 CHRNA1 (0.58) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL15007152 0.83 CHRNA1 (0.58) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL633367 0.83 CHRNA1 (0.58) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL8398736 0.81 PARP1 (0.58) PARP1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL4665718 0.81 CHRNA1 (0.56) PARP1CHRNA1CHRNGCHRNB1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1031941-C Process for preparing fluoroethylcamptothecin derivatives KYORIN SEIYAKU KK (JP) 1996-06-05 CN disclosed
EP-0471358-B1 Fluoroethylcamptothecin derivatives KYORIN SEIYAKU KK (JP) 1996-05-08 EP disclosed
EP-0325247-B1 CAMPTOTHECIN DERIVATIVES AND PROCESS FOR PREPARING SAME KABUSHIKI KAISHA YAKULT HONSHA (JP) 1993-05-19 EP disclosed
CN-1060095-A Fluoroethylcamptothederivatives derivatives KYORIN SEIYAKU KK (JP) 1992-04-08 CN disclosed
EP-0471358-A1 Fluoroethylcamptothecin derivatives KYORIN PHARMACEUTICAL CO., LTD. (JP) 1992-02-19 EP disclosed
US-5061800-A ANTITUMOR AGENTS KABUSHIKI KAISHA YAKULT HONSHA (JP) 1991-10-29 US disclosed
EP-0325247-A1 Camptothecin derivatives and process for preparing same KABUSHIKI KAISHA YAKULT HONSHA (JP) 1989-07-26 EP disclosed