SCHEMBL9047131

SCHEMBL9047131

CCCCC(=O)N1CC2(CCNCC2)c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.53
AKT1 P31749 5/20 0.49
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
USP2 O75604 1/20 0.41
BIRC2 Q13490 1/20 0.40
LTB4R2 Q9NPC1 2/20 0.39
SLC18A3 Q16572 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
P2RY1 P47900 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29644467 0.88 NOTUM (0.57) NOTUMAKT1ROCK2ROCK1BIRC2
SCHEMBL6543338 0.88 NOTUM (0.57) NOTUMAKT1ROCK2ROCK1BIRC2
SCHEMBL6543796 0.83 NOTUM (0.54) NOTUMAKT1ROCK2ROCK1BIRC2
SCHEMBL19750130 0.83 NOTUM (0.68) NOTUMAKT1HTR3EHTR3BHTR3A
SCHEMBL30232786 0.83 NOTUM (0.63) NOTUMAKT1ROCK2ROCK1HDAC1
SCHEMBL1572534 0.83 NOTUM (0.63) NOTUMAKT1ROCK2ROCK1HDAC1
SCHEMBL655024 0.81 NOTUM (0.80) NOTUMAKT1ROCK2ROCK1HDAC1
SCHEMBL6543487 0.81 NOTUM (0.55) NOTUMAKT1ROCK2ROCK1HDAC1
SCHEMBL1713780 0.81 NOTUM (0.57) NOTUMAKT1ROCK2ROCK1BIRC2
Hydrochloric Acid SCHEMBL2257588 0.80 NOTUM (0.78) NOTUMAKT1ROCK2ROCK1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702681-A1 SPIRO-SUBSTITUTED AZACYCLES AS NEUROKININ ANTAGONISTS MERCK & CO. INC. (US) 1996-03-27 EP disclosed
WO-1994029309-A1 SPIRO-SUBSTITUTED AZACYCLES AS NEUROKININ ANTAGONISTS MERCK & CO., INC. (US) 1994-12-22 WO disclosed