SCHEMBL9053133

SCHEMBL9053133

c1ccc2c(c1)CCc1c(N3CCNCC3)n[nH]c1-2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.60
HRH4 Q9H3N8 4/20 0.56
NPC1 O15118 1/20 0.42
KDR P35968 1/20 0.40
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
HTR7 P34969 2/20 0.39
HTR1A P08908 1/20 0.39
HTR2B P41595 1/20 0.39
HTR3A P46098 1/20 0.39
HTR6 P50406 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
RECQL P46063 1/20 0.39
KMT2A Q03164 1/20 0.39
PDGFRB P09619 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8000064 0.89 DRD4 (0.50) DRD4HRH4NPC1KDRHTR7
SCHEMBL8000470 0.81 DRD4 (0.66) DRD4HRH4KDRHRH2HRH1
SCHEMBL8009072 0.79 DRD4 (0.73) DRD4HRH4HRH2HRH1HRH3
SCHEMBL8018843 0.77 DRD4 (0.53) DRD4HRH4NPC1HRH2HRH1
SCHEMBL8009156 0.77 DRD4 (0.67) DRD4HRH4HRH2HRH1HRH3
SCHEMBL8009153 0.75 DRD4 (0.54) DRD4HRH4NPC1KDRHRH2
SCHEMBL8012111 0.75 DRD4 (1.00) DRD4HRH4NPC1KDRHRH2
Oxalic Acid SCHEMBL8011723 0.75 DRD4 (0.67) DRD4HRH4HRH2HRH1HRH3
SCHEMBL8015532 0.73 DRD4 (0.64) DRD4HRH4NPC1KDRHRH2
SCHEMBL605567 0.72 HRH4 (1.00) HRH4HRH2HRH1HRH3HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724572-A1 FUSED TRICYCLIC HETEROAROMATIC DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LTD. (GB) 1996-08-07 EP disclosed