SCHEMBL905395

SCHEMBL905395

Cc1ccccc1-c1cc(N2CCN(CC(=O)O)CC2)ncc1C(=O)N(C)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.82
GPBAR1 Q8TDU6 1/20 0.53
CYP3A4 P08684 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21235997 0.93 TACR1 (0.86) TACR1GPBAR1CYP3A4
SCHEMBL905355 0.91 TACR1 (0.77) TACR1GPBAR1CYP3A4
SCHEMBL905384 0.90 TACR1 (0.85) TACR1GPBAR1CYP3A4
SCHEMBL905333 0.90 TACR1 (0.85) TACR1GPBAR1CYP3A4
SCHEMBL7560214 0.90 TACR1 (0.84) TACR1GPBAR1CYP3A4
SCHEMBL29467378 0.90 TACR1 (1.00) TACR1GPBAR1
SCHEMBL905330 0.90 TACR1 (1.00) TACR1GPBAR1
SCHEMBL21235998 0.90 TACR1 (0.81) TACR1GPBAR1CYP3A4
SCHEMBL21141417 0.89 TACR1 (0.86) TACR1GPBAR1CYP3A4
Hydrochloric Acid SCHEMBL905341 0.89 TACR1 (0.98) TACR1GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1394150-B1 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists HOFFMANN LA ROCHE (CH) 2011-01-19 EP claimed