SCHEMBL905789

SCHEMBL905789

CC(C)(C)C(CCCCCCCCCCCCCCCC(=O)O)C(=O)OC(=N)CCC(=O)OC(=O)C(CCCCCCCCCCCCCCCC(=O)O)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 2/20 0.36
FFAR1 O14842 2/20 0.36
ALDH1A1 P00352 4/20 0.35
GSTK1 Q9Y2Q3 1/20 0.33
TSHR P16473 5/20 0.32
LMNA P02545 1/20 0.32
NFKB1 P19838 1/20 0.32
PMP22 Q01453 1/20 0.32
KDM4C Q9H3R0 2/20 0.32
KDM4A O75164 1/20 0.32
PHF8 Q9UPP1 1/20 0.32
KDM2A Q9Y2K7 1/20 0.32
PPARG P37231 6/20 0.32
PPARD Q03181 6/20 0.32
PPARA Q07869 6/20 0.32
GPR84 Q9NQS5 5/20 0.32
HDAC11 Q96DB2 5/20 0.32
TLR2 O60603 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
FABP4 P15090 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1509902 0.81 TSHR (0.35) FFAR4FFAR1ALDH1A1TSHRLMNA
SCHEMBL736106 0.76 FFAR4 (0.43) FFAR4FFAR1ALDH1A1GSTK1TSHR
SCHEMBL7905680 0.76 TSHR (0.40) TSHRSLC22A6
SCHEMBL1230057 0.72 TSHR (0.48) FFAR4FFAR1ALDH1A1TSHRLMNA
SCHEMBL20897216 0.72 FFAR4 (0.48) FFAR4FFAR1ALDH1A1GSTK1TSHR
SCHEMBL23611046 0.72 FFAR4 (0.48) FFAR4FFAR1ALDH1A1GSTK1TSHR
SCHEMBL905699 0.72 TSHR (0.48) FFAR4FFAR1ALDH1A1TSHRLMNA
SCHEMBL905720 0.72 TSHR (0.48) FFAR4FFAR1ALDH1A1TSHRLMNA
SCHEMBL379359 0.72 TSHR (0.48) FFAR4FFAR1ALDH1A1TSHRLMNA
SCHEMBL14119694 0.72 FFAR4 (0.48) FFAR4FFAR1ALDH1A1GSTK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2264065-B1 NOVEL INSULIN DERIVATIVES NOVO NORDISK AS (DK) 2017-03-08 EP disclosed
US-20140349925-A1 NOVEL INSULIN DERIVATIVES NOVO NORDISK AS (DK) 2014-11-27 US disclosed
US-8828923-B2 Insulin derivatives NOVO NORDISK A/S (DK) 2014-09-09 US disclosed
EP-2275439-B1 Novel insulin derivatives NOVO NORDISK AS (DK) 2014-03-26 EP disclosed
EP-2107069-B1 Novel insulin derivatives NOVO NORDISK AS (DK) 2013-01-16 EP disclosed
EP-2287184-A2 Novel insulin derivatives NOVO NORDISK A/S (DK) 2011-02-23 EP disclosed
EP-2275439-A2 Novel insulin derivatives NOVO NORDISK A/S (DK) 2011-01-19 EP disclosed
EP-2264065-A2 Novel Insulin Derivatives NOVO NORDISK A/S (DK) 2010-12-22 EP disclosed
EP-2264066-A2 Novel insulin derivatives NOVO NORDISK A/S (DK) 2010-12-22 EP disclosed
US-20100009899-A1 Novel Insulin Derivatives NOVO NORDISK A/S (DK) 2010-01-14 US disclosed
US-7615532-B2 Antidiabetic agents; insulin derivatives which are naturally occurring insulins or analogues thereof which have a side chain attached either to the alpha-amino group of the N-terminal amino acid residue of the B chain or to epsilon-amino group of a Lys residue present in the B chain of parent insulin NOVO NORDISK A/S (DE) 2009-11-10 US disclosed
EP-2107069-A2 Novel insulin derivatives NOVO NORDISK A/S (DK) 2009-10-07 EP disclosed
US-20060183668-A1 Antidiabetic agents; insulin derivatives which are naturally occurring insulins or analogues thereof which have a side chain attached either to the alpha-amino group of the N-terminal amino acid residue of the B chain or to epsilon-amino group of a Lys residue present in the B chain of parent insulin NOVO NORDISK A/S (DK) 2006-08-17 US disclosed
EP-1660531-A2 NOVEL INSULIN DERIVATIVES NOVO NORDISK A/S (DK) 2006-05-31 EP disclosed
WO-2005012347-A2 NOVEL INSULIN DERIVATIVES NOVO NORDISK A/S (DK) 2005-02-10 WO disclosed