SCHEMBL9060802

SCHEMBL9060802

O=[N+]([O-])c1ccc(CCCNCCO)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.64
CHRM2 P08172 1/20 0.59
KCNH2 Q12809 3/20 0.52
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
KCNJ1 P48048 2/20 0.48
ALDH1A1 P00352 2/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
NPC1 O15118 3/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
SLC22A2 O15244 1/20 0.46
ADRB1 P08588 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9194346 0.95 CHRM2 (0.62) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL9385011 0.94 TSHR (0.64) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL259753 0.90 TSHR (0.68) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL9450937 0.87 TSHR (0.64) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL5093330 0.85 CHRM2 (0.61) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL18067961 0.85 CHRM2 (0.60) TSHRCHRM2KCNH2MEN1KMT2A
Hydrochloric Acid SCHEMBL5099421 0.84 CHRM2 (0.59) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL8780911 0.84 CHRM2 (0.59) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL3118575 0.84 CHRM2 (0.59) TSHRCHRM2KCNH2MEN1KMT2A
SCHEMBL378397 0.83 TSHR (0.78) TSHRCHRM2KCNH2KCNJ1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3112948-A None JP disclosed
JP-8157429-A None JP disclosed
CN-105777559-A Synthesis method of nifekalant hydrochloride medical intermediate 2-[3-(4-nitrophenyl) propyl amino] ethyl alcohol 成都千叶龙华石油工程技术咨询有限公司 2016-07-20 CN disclosed
CN-105777559-A Synthesis method of nifekalant hydrochloride medical intermediate 2-[3-(4-nitrophenyl) propyl amino] ethyl alcohol 成都千叶龙华石油工程技术咨询有限公司 2016-07-20 CN disclosed
CN-103288751-B A kind of preparation method of high-purity nifekalant hydrochloride BAILI PHARMACEUTICAL CO., LTD., SICHUAN PROV. (CN) 2016-04-20 CN disclosed
CN-103288751-A Preparation method of high-purity nifekalant hydrochloride SICHUAN BIOKIN PHARMACEUTICAL CO LTD 2013-09-11 CN disclosed
JP-H08157429-A PRODUCTION OF N-(2-HYDROXYETHYL)-3-(4-NITROPHENYL) PROPYLAMINE MITSUI TOATSU CHEM INC 1996-06-18 JP disclosed
EP-0478268-B1 Polymerizable substituted amide compound, polymer obtained therefrom and nonlinear optical material using the same NIPPON PAINT CO LTD (JP) 1995-11-15 EP disclosed
EP-0369627-B1 Pyrimidinedione derivative compounds, method of producing the same and antiarrythmic agents containing the same MITSUI TOATSU CHEMICALS (JP) 1994-12-21 EP disclosed
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
US-5274061-A A 4-nitophenylaminoimido pendant group oriented by an electric field NIPPON PAINT CO., LTD. (JP) 1993-12-28 US disclosed
US-5200552-A POLYMERIZABLE SUBSTITUTED AMIDE COMPOUND, POLYMER OBTAINED THEREFROM AND NONLINEAR OPTICAL MATERIAL USING THE SAME NIPPON PAINT CO., LTD. (JP) 1993-04-06 US disclosed
EP-0478268-A1 Polymerizable substituted amide compound, polymer obtained therefrom and nonlinear optical material using the same Nippon Paint Co., Ltd. (JP) 1992-04-01 EP disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed
JP-H03112948-A N-(2-HYDROXYETHYL)-3-(4-NITROPHENYL)PROPYLAMINE AND PRODUCTION THEREOF MITSUI TOATSU CHEM INC 1991-05-14 JP disclosed
US-5008267-A Pyrimidinedione compounds, method of producing the same and antiarrythmic agents containing the same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1991-04-16 US disclosed
EP-0369627-A2 Pyrimidinedione derivative compounds, method of producing the same and antiarrythmic agents containing the same MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-05-23 EP disclosed