SCHEMBL9062175

SCHEMBL9062175

CCCc1cc(C(=O)O)ccc1OC(C(=O)NS(=O)(=O)c1ccc(C(=O)NO)cc1)c1ccc2c(c1)OCO2

nearest known ligand 0.85

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 16/20 0.85
EDNRB P24530 13/20 0.85
AGTR1 P30556 3/20 0.53
AGTR2 P50052 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341739 0.92 EDNRA (0.88) EDNRAEDNRBAGTR1AGTR2
L-754142 SCHEMBL29551244 0.92 EDNRA (1.00) EDNRAEDNRBAGTR1AGTR2
L-754142 SCHEMBL4193035 0.92 EDNRA (1.00) EDNRAEDNRBAGTR1AGTR2
SCHEMBL7339397 0.92 EDNRA (0.88) EDNRAEDNRBAGTR1AGTR2
SCHEMBL7338764 0.91 EDNRA (0.84) EDNRAEDNRBAGTR1AGTR2
SCHEMBL7337876 0.91 EDNRA (0.89) EDNRAEDNRBAGTR1AGTR2
L-754142 SCHEMBL7722258 0.91 EDNRA (0.98) EDNRAEDNRBAGTR1AGTR2
L-754142 SCHEMBL4202655 0.91 EDNRA (0.98) EDNRAEDNRBAGTR1AGTR2
SCHEMBL7333156 0.91 EDNRA (0.85) EDNRAEDNRBAGTR1AGTR2
SCHEMBL7338714 0.91 EDNRA (0.85) EDNRAEDNRBAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996009818-A1 ENDOTHELIN RECEPTOR ANTAGONISTS FOR THE TREATMENT OF EMESIS MERCK & CO., INC. (US) 1996-04-04 WO claimed