SCHEMBL9070856

SCHEMBL9070856

COC[C@@H](C)Oc1cc(C(=O)Nc2ccc(C(=O)O)cn2)cc(Oc2cc(F)cc(Cl)c2)n1

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GCK P35557 20/20 0.72
RARG P13631 1/20 0.72
RARA P10276 1/20 0.57
RARB P10826 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9071063 0.94 GCK (0.80) GCKRARGRARARARB
SCHEMBL5653831 0.90 GCK (0.88) GCKRARGRARARARB
SCHEMBL9071047 0.90 GCK (0.58) GCKRARGRARARARB
SCHEMBL2667576 0.89 GCK (0.71) GCKRARGRARARARB
SCHEMBL9070859 0.89 GCK (0.57) GCKRARGRARARARB
SCHEMBL2667803 0.88 GCK (0.80) GCKRARGRARARARB
SCHEMBL9071029 0.85 GCK (0.78) GCKRARGRARARARB
SCHEMBL9071059 0.85 GCK (0.51) GCKRARG
SCHEMBL5652615 0.84 GCK (1.00) GCKRARGRARARARB
SCHEMBL14366905 0.83 GCK (0.77) GCKRARGRARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009083553-A1 AZINE COMPOUNDS AS GLUCOKINASE ACTIVATORS RHEOSCIENCE A/S (DK) 2009-07-09 WO disclosed