SCHEMBL9074014

SCHEMBL9074014

NC[C@H]1CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)O

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACE P12821 8/20 0.50
ACE2 Q9BYF1 6/20 0.50
ATM Q13315 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
ALDH1A1 P00352 1/20 0.48
HSD17B10 Q99714 1/20 0.48
F2 P00734 1/20 0.48
PRSS1 P07477 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9074016 1.00 ACE (0.50) ACEACE2ATML3MBTL1ALDH1A1
SCHEMBL9076967 0.85 ACE2 (0.45) ACEACE2ATML3MBTL1F2
SCHEMBL9076970 0.85 ACE2 (0.45) ACEACE2ATML3MBTL1F2
SCHEMBL9074952 0.84 ACE2 (0.46) ACEACE2ATML3MBTL1F2
SCHEMBL9074948 0.84 ACE2 (0.46) ACEACE2ATML3MBTL1F2
SCHEMBL7342855 0.83 F2 (0.46) ACEACE2ATML3MBTL1F2
SCHEMBL9076347 0.83 F2 (0.46) ACEACE2ATML3MBTL1F2
SCHEMBL9074561 0.82 ACE2 (0.42) ACEACE2ATML3MBTL1F2
SCHEMBL9074564 0.82 ACE2 (0.42) ACEACE2ATML3MBTL1F2
SCHEMBL18064472 0.81 ACE (0.53) ACEACE2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0623596-A1 N-acylpyrrolidines or N-acylpiperidines having a guanidinyl- or amidinyl-substituted side chain as thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-11-09 EP disclosed