SCHEMBL9075795

SCHEMBL9075795

O=C(O)C(O)(c1ccccc1)c1ccc(Br)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.64
CYP2D6 P10635 1/20 0.50
HIF1A Q16665 1/20 0.50
KIF11 P52732 1/20 0.45
CYP1A2 P05177 1/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
ALDH1A1 P00352 3/20 0.40
AKR1C3 P42330 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9076491 1.00 CYP2C9 (0.64) CYP2C9CYP2D6HIF1AKIF11CYP1A2
SCHEMBL9076924 1.00 CYP2C9 (0.64) CYP2C9CYP2D6HIF1AKIF11CYP1A2
SCHEMBL3172975 0.94 CYP2C9 (0.59) CYP2C9CYP2D6HIF1AKIF11CYP1A2
Benzylic Acid SCHEMBL7066 0.87 CYP2C9 (0.74) CYP2C9CYP2D6HIF1ACYP1A2ALDH1A1
Benzylic Acid SCHEMBL4823051 0.85 CYP2C9 (0.65) CYP2C9CYP2D6HIF1ACYP1A2ALDH1A1
Benzylic Acid SCHEMBL1680669 0.84 CYP2C9 (0.71) CYP2C9CYP2D6HIF1ACYP1A2ALDH1A1
Benzylic Acid SCHEMBL9568239 0.84 CYP2C9 (0.71) CYP2C9CYP2D6HIF1ACYP1A2ALDH1A1
Benzylic Acid SCHEMBL9181980 0.84 CYP2C9 (0.71) CYP2C9CYP2D6HIF1ACYP1A2ALDH1A1
Benzylic Acid SCHEMBL20957595 0.84 CYP2C9 (0.71) CYP2C9CYP2D6HIF1ACYP1A2ALDH1A1
Benzylic Acid SCHEMBL11049826 0.84 CYP2C9 (0.71) CYP2C9CYP2D6HIF1ACYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5569447-A TOMOGRAPHIC IMAGING AGENTS THE UNITED STATES OF AMERICA REPRESENTED BY THE SECRETARY DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1996-10-29 US disclosed
US-5387409-A Diagnostic imaging agents, e.g. hypoxic tissue; radiotherapy; kits BRACCO INTERNATIONAL B.V. (NL) 1995-02-07 US disclosed
EP-0441491-A1 Boronic acid adducts of rhenium dioxime and technetium-99M dioxime complexes containing a biochemically active group BRACCO INTERNATIONAL B.V. (NL) 1991-08-14 EP disclosed