SCHEMBL9078296

SCHEMBL9078296

NC1CC(c2c[nH]c3ccc(Cn4cncn4)cc23)C1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 16/20 0.53
HTR1B P28222 16/20 0.53
HTR1A P08908 1/20 0.53
ADRA2C P18825 1/20 0.53
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
HRH1 P35367 1/20 0.53
HTR2B P41595 1/20 0.53
SLC6A4 P31645 1/20 0.41
CYP19A1 P11511 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9076100 0.86 HTR1B (0.61) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL9076096 0.86 HTR1B (0.61) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL9077368 0.86 HTR1B (0.61) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL7822979 0.84 HTR1D (0.56) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL8784217 0.84 HTR1D (0.53) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL8784664 0.83 HTR1D (0.55) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL8784644 0.81 HTR1D (0.53) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL9274399 0.78 HTR1D (0.53) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL7839523 0.74 HTR1D (0.73) HTR1DHTR1BHTR1AADRA2CHTR2A
SCHEMBL7479049 0.74 HTR1D (0.69) HTR1DHTR1BHTR1AADRA2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5567726-A SELECTIVE AGONISTS OF 5-HYDROXYTRYPTAMINE-LIKE RECEPTORS; USEFUL IN TREATMENT OF MIGRAINE AND ASSOCIATED DISORDERS MERCK, SHARP & DOHME LTD. (GB) 1996-10-22 US disclosed
WO-1994002477-A1 IMIDAZOLE, TRIAZOLE AND TETRAZOLE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1994-02-03 WO disclosed