SCHEMBL9079477

SCHEMBL9079477

CC(O)=C(C#N)C(=O)Nc1ccc(O)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 11/20 0.74
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
ALDH1A1 P00352 4/20 0.53
CYP3A4 P08684 2/20 0.53
TSHR P16473 2/20 0.53
CA12 O43570 1/20 0.53
BRD4 O60885 1/20 0.53
NR1I2 O75469 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
MB P02144 1/20 0.53
CYP1A1 P04798 1/20 0.53
CA3 P07451 1/20 0.53
MAPT P10636 1/20 0.53
RARG P13631 1/20 0.53
ALOX5AP P20292 1/20 0.53
CA4 P22748 1/20 0.53
CA7 P43166 1/20 0.53
NR1I3 Q14994 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8810371 1.00 DHODH (0.74) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL13531076 0.88 DHODH (0.72) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL12202668 0.88 DHODH (0.72) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL3250475 0.88 DHODH (0.82) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL3250476 0.88 DHODH (0.82) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL5914902 0.88 DHODH (0.82) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL5914890 0.87 DHODH (0.70) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL5914911 0.87 DHODH (0.71) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL5914889 0.87 DHODH (0.70) DHODHMEN1KMT2AALDH1A1CYP3A4
SCHEMBL5914891 0.87 DHODH (0.70) DHODHMEN1KMT2AALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532259-A ANTITUMOR HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-02 US disclosed
US-5494911-A TREATING LEUKEMIA, SARCOMA, CARCINOMA, LYMPHOMA, SKIN CANCER HOECHST AKTIENGESELLSCHAFT (DE) 1996-02-27 US disclosed