SCHEMBL9099759

SCHEMBL9099759

CNc1nc(N)nc2c1CN(S(C)(=O)=O)CC2

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.40
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KCNH2 Q12809 4/20 0.34
PIK3R1 P27986 2/20 0.34
PIK3CA P42336 2/20 0.34
F12 P00748 1/20 0.34
GPR6 P46095 2/20 0.33
PDE10A Q9Y233 1/20 0.33
CNR2 P34972 2/20 0.33
HTR6 P50406 1/20 0.32
HRH4 Q9H3N8 3/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2249696 0.69 PDGFRB (0.47) NPC1RAB9APIK3R1PIK3CAPIK3CD
SCHEMBL4990795 0.63 NPC1 (0.39) NPC1RAB9AF12CNR2
SCHEMBL23921753 0.63 NPC1 (0.38) NPC1RAB9AF12PDE10ACNR2
SCHEMBL22702917 0.62 F12 (0.46) F12
SCHEMBL22492312 0.62 F12 (0.39) NPC1RAB9AF12
SCHEMBL4982872 0.61 NPC1 (0.39) NPC1RAB9AF12
SCHEMBL19493556 0.60 ESR1 (0.44) CYP2C19NPC1RAB9AF12CNR2
SCHEMBL12680946 0.60 NPC1 (0.60) NPC1RAB9APDE10ACNR2
SCHEMBL2915641 0.59 F12 (0.38) NPC1RAB9AF12
SCHEMBL23921754 0.59 KCNK3 (0.35) NPC1RAB9AF12GPR6PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2459197-A1 COMPOUNDS FOR THE REDUCTION OF -AMYLOID PRODUCTION Bristol-Myers Squibb Company (US) 2012-06-06 EP claimed