SCHEMBL9118070

SCHEMBL9118070

C[C@H]([C@](O)(Cn1ccnc1)c1ccc(F)cc1F)S(=O)(=O)N(C)Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 12/20 0.53
CYP2C9 P11712 4/20 0.36
CYP2C19 P33261 4/20 0.36
CYP2B6 P20813 1/20 0.36
CYP3A5 P20815 1/20 0.36
CYP3A7 P24462 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP3A43 Q9HB55 1/20 0.36
CYP46A1 Q9Y6A2 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 3/20 0.35
CYP2D6 P10635 3/20 0.35
PTGS2 P35354 1/20 0.35
HMOX1 P09601 1/20 0.33
CYP19A1 P11511 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9121589 0.85 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9119273 0.85 CYP3A4 (0.62) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9119197 0.75 CYP3A4 (0.54) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9119129 0.75 CYP3A4 (0.56) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9045971 0.75 CYP3A4 (0.69) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL8341941 0.74 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9044673 0.74 CYP3A4 (0.67) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9120293 0.73 CYP3A4 (0.66) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9122089 0.73 CYP3A4 (0.55) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5
SCHEMBL9117376 0.72 CYP3A4 (0.60) CYP3A4CYP2C9CYP2C19CYP2B6CYP3A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389663-A Fungicides TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0510700-A2 Azole compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-10-28 EP disclosed