SCHEMBL9126409

SCHEMBL9126409

COc1cc2c(c(O)c1OC)C(Cc1ccc(F)cc1)NCC2

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 3/20 0.64
BCHE P06276 1/20 0.56
ADRB2 P07550 2/20 0.54
ADRB1 P08588 2/20 0.54
ADRB3 P13945 2/20 0.54
KDM4E B2RXH2 1/20 0.54
MAPT P10636 1/20 0.54
PKM P14618 1/20 0.54
HTR1A P08908 1/20 0.53
ADRA2A P08913 1/20 0.53
DRD1 P21728 1/20 0.53
PTGS1 P23219 1/20 0.53
OPRM1 P35372 1/20 0.53
DRD3 P35462 1/20 0.53
DHFR P00374 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558905 0.90 TBXA2R (0.59) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL8982767 0.89 TBXA2R (0.63) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL8982937 0.87 TBXA2R (0.73) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL8982846 0.84 TBXA2R (0.63) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL8983089 0.83 TBXA2R (0.57) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL8982824 0.83 TBXA2R (0.53) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL8982857 0.81 TBXA2R (0.54) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL6393104 0.81 KDM4C (0.51) TBXA2RBCHEKDM4EMAPTPKM
SCHEMBL8982983 0.79 TBXA2R (0.52) TBXA2RBCHEADRB2ADRB1ADRB3
SCHEMBL27617352 0.79 KDM4E (0.54) TBXA2RBCHEADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446164-A Regioselective cyclization of phenethylamide derivative in presence of phosphoric acid halide, reducing formed compound BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-29 US disclosed