SCHEMBL9129554

SCHEMBL9129554

COc1cc(C=CCCBr)cc(OC)c1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP1B1 Q16678 1/20 0.53
TUBB1 Q9H4B7 15/20 0.53
TUBB4A P04350 10/20 0.53
TUBB P07437 10/20 0.53
TUBA3C P0DPH7 10/20 0.53
TUBA1B P68363 10/20 0.53
TUBA4A P68366 10/20 0.53
TUBB4B P68371 10/20 0.53
TUBB3 Q13509 10/20 0.53
TUBB2A Q13885 10/20 0.53
TUBB8 Q3ZCM7 10/20 0.53
TUBA3E Q6PEY2 10/20 0.53
TUBA1A Q71U36 10/20 0.53
TUBA1C Q9BQE3 10/20 0.53
TUBB6 Q9BUF5 10/20 0.53
TUBB2B Q9BVA1 10/20 0.53
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9129548 1.00 CYP1A1 (0.53) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL8627361 0.90 TUBB1 (0.50) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL4765514 0.90 TUBB1 (0.50) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL4765528 0.90 TUBB1 (0.50) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL4450715 0.85 CYP1A1 (0.56) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL4450716 0.85 CYP1A1 (0.56) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL29565593 0.85 CYP1A1 (0.56) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL9763608 0.82 TUBB1 (0.55) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL5691704 0.82 CYP1A1 (0.53) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A
SCHEMBL9763615 0.82 TUBB1 (0.55) CYP1A1CYP1A2CYP1B1TUBB1TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0541798-B1 NEW DIAMINE COMPOUND AND BRAIN PROTECTING AGENT CONTAINING THE SAME KOWA CO (JP) 1995-11-29 EP disclosed
US-5389630-A Diamine compound and brain protecting agent containing the same KOWA CO., LTD. (JP) 1995-02-14 US disclosed
EP-0541798-A1 NEW DIAMINE COMPOUND AND BRAIN PROTECTING AGENT CONTAINING THE SAME Kowa Company Ltd. (JP) 1993-05-19 EP disclosed