SCHEMBL9130576

SCHEMBL9130576

NNC(=O)Cc1ccc2c(c1)NC(=O)CO2

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.60
ALDH1A1 P00352 4/20 0.52
MAPT P10636 3/20 0.52
TSHR P16473 1/20 0.51
MMP12 P39900 1/20 0.50
NR3C2 P08235 2/20 0.49
GAA P10253 1/20 0.49
KDM4E B2RXH2 1/20 0.48
KMT2A Q03164 1/20 0.47
SMYD3 Q9H7B4 1/20 0.47
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47
DRD3 P35462 1/20 0.47
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2068664 0.93 PARP1 (0.55) PARP1ALDH1A1MAPTTSHRMMP12
Hydrochloric Acid SCHEMBL1433215 0.92 PARP1 (0.54) PARP1ALDH1A1MAPTTSHRMMP12
SCHEMBL14073116 0.86 PARP1 (0.62) PARP1ALDH1A1MAPTTSHRMMP12
SCHEMBL16421393 0.85 PARP1 (0.65) PARP1ALDH1A1MAPTTSHRMMP12
SCHEMBL14073095 0.85 MAPT (0.60) PARP1ALDH1A1MAPTTSHRKMT2A
SCHEMBL4286655 0.83 PARP1 (0.67) PARP1ALDH1A1MAPTTSHRMMP12
SCHEMBL10923540 0.82 PARP1 (0.69) PARP1ALDH1A1MAPTTSHRMMP12
SCHEMBL4295364 0.82 PARP1 (0.65) PARP1ALDH1A1MAPTTSHRMMP12
SCHEMBL14073059 0.82 GAA (0.59) PARP1ALDH1A1MAPTGAASMYD3
SCHEMBL14073688 0.82 PARP1 (0.54) PARP1ALDH1A1MAPTTSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1121072-A Acetamides MERCK PATENG GES MIT BESCHRANK (DE) 1996-04-24 CN disclosed
US-5472961-A Acetamides MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-12-05 US disclosed