SCHEMBL9130912

SCHEMBL9130912

CCCCc1nc2ccc(N)cc2c(=O)[nH]1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.66
MAPT P10636 4/20 0.51
PKM P14618 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
ALDH1A1 P00352 2/20 0.49
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47
TUBA4A P68366 1/20 0.47
TUBB4B P68371 1/20 0.47
TUBB3 Q13509 1/20 0.47
TUBB2A Q13885 1/20 0.47
TUBB8 Q3ZCM7 1/20 0.47
TUBA3E Q6PEY2 1/20 0.47
TUBA1A Q71U36 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9129643 0.92 KDM4C (0.56) PARP1MAPTPKMKDM4EMEN1
SCHEMBL9131594 0.85 TNKS2 (0.62) PARP1MAPTPKMKDM4EMEN1
SCHEMBL7418316 0.84 PARP1 (0.68) PARP1MAPTKMT2AALDH1A1TUBB4A
SCHEMBL9327417 0.83 PARP1 (0.66) PARP1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL13111952 0.83 PARP1 (0.66) PARP1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL7415916 0.81 PARP1 (0.63) PARP1MAPTKDM4ETUBB4ATUBB
SCHEMBL11376990 0.81 PARP1 (0.63) PARP1MAPTKDM4EMEN1KMT2A
SCHEMBL9376967 0.81 PARP1 (0.63) PARP1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8805356 0.80 MAPT (0.79) MAPTPKMKDM4EMEN1KMT2A
SCHEMBL168776 0.80 PARP1 (1.00) PARP1MEN1KMT2ATNKS2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441959-A Hypotensive agents; treating congestive heart failure and glaucoma,inhibiting restenosis MERCK & CO., INC. (US) 1995-08-15 US disclosed