SCHEMBL9136458

SCHEMBL9136458

CC(=O)CNc1ccc(N)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.48
MAPT P10636 2/20 0.48
ESR1 P03372 2/20 0.47
CYP19A1 P11511 2/20 0.47
ESR2 Q92731 2/20 0.47
PKM P14618 2/20 0.44
CYP2C19 P33261 2/20 0.44
TDP1 Q9NUW8 3/20 0.44
MEN1 O00255 2/20 0.44
LMNA P02545 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
APEX1 P27695 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.40
TSHR P16473 2/20 0.40
DHFR P00374 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HIF1A Q16665 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40
SLC22A8 Q8TCC7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28003608 0.83 CYP19A1 (0.42) RAB9AMAPTESR1CYP19A1ESR2
SCHEMBL9419326 0.81 MAPT (0.54) RAB9AMAPTTDP1MEN1KMT2A
SCHEMBL3995569 0.81 ESR1 (0.55) RAB9AMAPTESR1CYP19A1ESR2
SCHEMBL12378828 0.81 MEN1 (0.52) RAB9AMAPTMEN1LMNAKMT2A
SCHEMBL1312570 0.81 MAPT (0.55) RAB9AMAPTESR1CYP19A1ESR2
Hydrochloric Acid SCHEMBL11148769 0.81 MAPT (0.55) RAB9AMAPTESR1CYP19A1ESR2
Hydrochloric Acid SCHEMBL7148684 0.81 MAPT (0.55) RAB9AMAPTESR1CYP19A1ESR2
SCHEMBL4582345 0.81 MAPT (0.54) RAB9AMAPTTDP1MEN1LMNA
SCHEMBL8487007 0.80 CA12 (0.46) RAB9AMAPTESR1CYP19A1ESR2
SCHEMBL13773412 0.80 CA12 (0.49) RAB9AMAPTTDP1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773768-B1 PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS EXELIXIS INC (US) 2018-08-22 EP disclosed
US-5453501-A Phthalocyanine reactive dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1995-09-26 US disclosed
EP-0582886-A1 Phthalocyanine reactive dyes BAYER AG (DE) 1994-02-16 EP disclosed
EP-0038453-B1 PROCESS FOR THE PREPARATION OF WATER SOLUBLE PHTHALOCYANINE DYESTUFFS BAYER AG (DE) 1983-05-25 EP disclosed
EP-0012349-B1 PROCESS FOR PRODUCING PHTHALOCYANINE REACTIVE DYESTUFFS BAYER AG (DE) 1981-11-04 EP disclosed
EP-0038453-A2 Process for the preparation of water soluble phthalocyanine dyestuffs BAYER AG (DE) 1981-10-28 EP disclosed
US-4246174-A Process for the preparation of phthalocyanine reactive dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1981-01-20 US disclosed
EP-0012349-A2 Process for producing phthalocyanine reactive dyestuffs BAYER AG (DE) 1980-06-25 EP disclosed