SCHEMBL9145502

SCHEMBL9145502

O=C(O)c1cn2c3c(c(Cl)ccc3c1=O)CCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 2/20 0.40
CSNK2B P67870 2/20 0.40
CSNK2A1 P68400 2/20 0.40
BCL2 P10415 1/20 0.39
BCL2L1 Q07817 1/20 0.39
MCL1 Q07820 1/20 0.39
TSHR P16473 2/20 0.37
POLB P06746 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36
KDM4E B2RXH2 6/20 0.35
ALDH1A1 P00352 2/20 0.35
HSP90AA1 P07900 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ADRA2B P18089 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11163715 0.93 CSNK2A2 (0.41) CSNK2A2CSNK2BCSNK2A1BCL2BCL2L1
SCHEMBL10903433 0.81 CHRM1 (0.39) TSHRPOLBKDM4EALDH1A1HSP90AA1
SCHEMBL10905876 0.79 HSD17B10 (0.40) POLBKDM4EALDH1A1HSP90AA1RXFP1
SCHEMBL10998660 0.78 TSHR (0.39) CSNK2A2CSNK2BCSNK2A1BCL2BCL2L1
SCHEMBL9031451 0.78 CSNK2A2 (0.40) CSNK2A2CSNK2BCSNK2A1BCL2BCL2L1
SCHEMBL11163211 0.78 KDM4E (0.47) POLBKMT2AMEN1KDM4EALDH1A1
SCHEMBL10940721 0.78 KDM4E (0.44) TSHRPOLBKDM4EALDH1A1HSP90AA1
SCHEMBL10998820 0.77 KDM4E (0.55) CSNK2A2CSNK2BCSNK2A1POLBKMT2A
Hydrochloric Acid SCHEMBL11160600 0.77 KDM4E (0.45) TSHRPOLBKDM4EALDH1A1HSP90AA1
SCHEMBL11175761 0.77 KDM4E (0.33) TSHRPOLBKMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5457104-A Antibacterials BAYER AKTIENGESELLSCHAFT (DE) 1995-10-10 US disclosed
US-4416884-A ANTIBIOTIC, BACTERICIDE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1983-11-22 US disclosed
US-4317820-A β-Lactam series compound and antibacterial pharmaceutical composition containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1982-03-02 US disclosed