SCHEMBL9160121

SCHEMBL9160121

COc1ccc(CN2CCN(C(=O)[C@@H](C)N)CC2)c(OC)c1OC

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.71
KDM4E B2RXH2 3/20 0.59
ALDH1A1 P00352 2/20 0.59
HTT P42858 2/20 0.59
PKM P14618 1/20 0.59
MEN1 O00255 4/20 0.58
KMT2A Q03164 4/20 0.58
CHRM2 P08172 2/20 0.55
OPRK1 P41145 2/20 0.55
CYP1A2 P05177 1/20 0.55
SLC6A4 P31645 1/20 0.55
OPRD1 P41143 1/20 0.55
APOBEC3A P31941 1/20 0.54
CTDSP1 Q9GZU7 1/20 0.54
APOBEC3G Q9HC16 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.53
LMNA P02545 2/20 0.52
ADORA3 P0DMS8 1/20 0.52
CHRM1 P11229 1/20 0.52
DRD2 P14416 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9158845 1.00 CYP2C19 (0.71) CYP2C19KDM4EALDH1A1HTTPKM
Hydrochloric Acid SCHEMBL9426145 0.99 CYP2C19 (0.69) CYP2C19KDM4EALDH1A1HTTPKM
Hydrochloric Acid SCHEMBL9426011 0.99 CYP2C19 (0.69) CYP2C19KDM4EALDH1A1HTTPKM
SCHEMBL9425561 0.91 CYP2C19 (0.68) CYP2C19KDM4EALDH1A1HTTPKM
SCHEMBL10858979 0.89 CYP2C19 (0.69) CYP2C19KDM4EALDH1A1HTTPKM
SCHEMBL10858976 0.89 CYP2C19 (0.69) CYP2C19KDM4EALDH1A1HTTPKM
Hydrochloric Acid SCHEMBL10859968 0.88 CYP2C19 (0.67) CYP2C19KDM4EALDH1A1HTTPKM
Hydrochloric Acid SCHEMBL10859963 0.88 CYP2C19 (0.67) CYP2C19KDM4EALDH1A1HTTPKM
SCHEMBL9152616 0.86 CYP2C19 (0.62) CYP2C19KDM4EALDH1A1HTTPKM
SCHEMBL9154894 0.85 CYP2C19 (0.61) CYP2C19KDM4EALDH1A1HTTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0533516-B1 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-02-08 EP disclosed
US-5340809-A Antihypoxic, antiischemic agents ADIR ET COMPAGNIE (FR) 1994-08-23 US disclosed
EP-0533516-A2 Amides of 1-(alkoxybenzyl)piperazines, processes for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-03-24 EP disclosed