SCHEMBL9163382

SCHEMBL9163382

C[C@@H]1CN(Cc2ccccc2Br)C[C@@H](C)O1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.67
HTT P42858 1/20 0.67
CYP2A13 Q16696 2/20 0.59
TDP1 Q9NUW8 2/20 0.51
ALDH1A1 P00352 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
ATM Q13315 1/20 0.47
TSHR P16473 1/20 0.47
RECQL P46063 1/20 0.47
FAAH O00519 1/20 0.43
LMNA P02545 2/20 0.42
GAA P10253 2/20 0.42
SLC2A1 P11166 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
HTR6 P50406 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9161601 1.00 KDM4E (0.67) KDM4EHTTCYP2A13TDP1ALDH1A1
SCHEMBL9390972 1.00 KDM4E (0.67) KDM4EHTTCYP2A13TDP1ALDH1A1
SCHEMBL22711519 0.80 KDM4E (0.67) KDM4EHTTCYP2A13TDP1ALDH1A1
SCHEMBL7372983 0.80 KDM4E (1.00) KDM4EHTTCYP2A13TDP1ALDH1A1
SCHEMBL1591865 0.75 KDM4E (0.65) KDM4EHTTCYP2A13TDP1LMNA
SCHEMBL70870 0.75 KDM4E (0.65) KDM4EHTTCYP2A13TDP1LMNA
SCHEMBL4510409 0.75 KDM4E (0.65) KDM4EHTTCYP2A13TDP1LMNA
SCHEMBL1591329 0.75 KDM4E (0.65) KDM4EHTTCYP2A13TDP1LMNA
SCHEMBL31193156 0.75 KDM4E (0.60) KDM4EHTTCYP2A13TDP1ALDH1A1
SCHEMBL13850015 0.74 CYP2A13 (1.00) KDM4EHTTCYP2A13TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5382666-A Heterocyclic intermediates ORTHO PHARMACEUTICAL CORPORATION (US) 1995-01-17 US disclosed
WO-1994015926-A1 ANGIOTENSIN II INHIBITORS ORTHO PHARMACEUTICAL CORPORATION (US) 1994-07-21 WO disclosed
US-5256658-A Biphenylyl tetrazoles for hypertension in mammals ORTHO PHARMACEUTICAL CORPORATION (US) 1993-10-26 US disclosed