SCHEMBL9163473

SCHEMBL9163473

COC(=S)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.48
MAPT P10636 3/20 0.48
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
ALDH1A1 P00352 3/20 0.45
LMNA P02545 2/20 0.45
GAA P10253 2/20 0.45
EGFR P00533 1/20 0.45
ALOX12 P18054 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PDCD1 Q15116 1/20 0.44
CD274 Q9NZQ7 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
WDR5 P61964 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HTT P42858 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL812710 0.86 TSHR (0.52) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
Thiobenzoic Acid SCHEMBL2320796 0.80 HPGD (0.47) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
SCHEMBL10649450 0.80 PLAU (0.53) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL1479349 0.78 SMN1; SMN2 (0.43) SMN1; SMN2MAPTNPC1RAB9ACTDSP1
SCHEMBL31090739 0.78 KCNN4 (0.41) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
SCHEMBL9167776 0.77 EGFR (0.56) SMN1; SMN2ALDH1A1EGFRNCOA3
Thiobenzoic Acid SCHEMBL10902274 0.77 HPGD (0.44) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
Thiobenzoic Acid SCHEMBL9789964 0.76 ESR1 (0.44) MAPTNPC1RAB9AALDH1A1LMNA
SCHEMBL9166737 0.76 ESR2 (0.51) SMN1; SMN2ALDH1A1LMNAEGFRL3MBTL1
SCHEMBL11665324 0.76 EGFR (0.44) SMN1; SMN2MAPTNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269859-B2 Pyrazolotriazine compounds OTSUKA PHARMA CO LTD (JP) 1995-10-18 EP disclosed
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed
US-4824834-A TREATING GOUT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-04-25 US disclosed
EP-0269859-A2 Pyrazolotriazine compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-06-08 EP disclosed