SCHEMBL9164057

SCHEMBL9164057

O=C1CCc2cc(OCCCBr)ccc2N1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 17/20 0.68
MAOA P21397 16/20 0.68
PDE3B Q13370 2/20 0.55
PDE3A Q14432 2/20 0.55
HTR1A P08908 1/20 0.55
DRD2 P14416 1/20 0.55
DRD4 P21917 1/20 0.55
HTR2A P28223 1/20 0.55
HTR2C P28335 1/20 0.55
SLC6A4 P31645 1/20 0.55
HTR7 P34969 1/20 0.55
DRD3 P35462 1/20 0.55
MEN1 O00255 1/20 0.51
ABCC4 O15439 1/20 0.51
CACNA1F O60840 1/20 0.51
ABCB11 O95342 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1036438 0.96 MAOB (0.67) MAOBMAOAPDE3BPDE3AHTR1A
SCHEMBL11276922 0.94 MAOB (0.65) MAOBMAOAPDE3BPDE3AHTR1A
SCHEMBL11273468 0.94 MAOB (0.65) MAOBMAOAPDE3BPDE3AHTR1A
SCHEMBL25362567 0.93 MAOB (0.67) MAOBMAOAPDE3BPDE3AHTR1A
SCHEMBL252282 0.89 MAOB (0.70) MAOBMAOA
SCHEMBL30546591 0.89 MAOB (0.70) MAOBMAOA
SCHEMBL12359302 0.87 MAOB (0.70) MAOBMAOAPDE3BPDE3AHTR1A
SCHEMBL426467 0.87 MAOB (0.70) MAOBMAOAPDE3BPDE3AHTR1A
SCHEMBL10675306 0.86 MAOB (0.68) MAOBMAOAPDE3BPDE3AHTR1A
SCHEMBL6585538 0.86 MAOB (0.68) MAOBMAOAPDE3BPDE3AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025229046-A1 SUBSTITUTED HYDROQUINOLINES FOR THE TREATMENT OF GLIOBLASTOMA MULTIFORME MOLIUS SAGLIK TEKNOLOJILERI ANONIM SIRKETI (TR) 2025-11-06 WO disclosed
EP-4644375-A1 SUBSTITUTED HYDROQUINOLINES FOR THE TREATMENT OF GLIOBLASTOMA MULTIFORME Molius Saglik Teknolojileri Anonim Sirketi (TR) 2025-11-05 EP disclosed
US-5434164-A Carbostyril derivatives and salts thereof and pharmaceutical compositions for inhibiting adhesion of thrombocytes OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1995-07-18 US disclosed
EP-0240015-B1 Carbostyril derivatives, process for preparing them, pharmaceutical composition, and use OTSUKA PHARMA CO LTD (JP) 1994-12-28 EP disclosed
US-5008274-A Carbostyril derivatives and salts thereof and pharmaceutical composition for inhibiting adhesion of thrombocytes OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-04-16 US disclosed
US-4918073-A CALCIUM ANTAGONISTS HOECHST AKTIENGESELLSCHAFT (DE) 1990-04-17 US disclosed
US-4746661-A Phenylpiperazine propyloxyquinolinones and methods for sedating and inhibiting aggression in livestock therewith HOECHST AKTIENGESELLSCHAFT (DE) 1988-05-24 US disclosed
EP-0240015-A2 Carbostyril derivatives, process for preparing them, pharmaceutical composition, and use OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-10-07 EP disclosed
EP-0229623-A2 Diaryl-substituted alkylamines, procedure for their preparation, their application and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1987-07-22 EP disclosed
EP-0182247-A1 Substituted phenyl piperazine derivatives, processes for their preparation and the use of substituted phenyl piperazine derivatives as aggression inhibitors in animals HOECHST AKTIENGESELLSCHAFT (DE) 1986-05-28 EP disclosed
EP-0003771-B1 CARBOSTYRILE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1982-10-20 EP disclosed
US-4329347-A Cardiotonic and antithrombotic sulfur-containing derivatives of carbostyril BOEHRINGER INGELHEIM GMBH (DE) 1982-05-11 US disclosed
EP-0005828-B1 NEW SUBSTITUTED PHENYLPIPERAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION HOECHST AKTIENGESELLSCHAFT (DE) 1981-03-11 EP disclosed
US-4234584-A NEUROLEPTIC HOECHST AKTIENGESELLSCHAFT (DE) 1980-11-18 US disclosed
EP-0003771-A1 Carbostyrile derivatives, their preparation and pharmaceutical compositions containing them Dr. Karl Thomae GmbH (DE) 1979-09-05 EP disclosed