SCHEMBL9178373

SCHEMBL9178373

COC(=O)C(C)(C)Cc1c(SC(C)(C)C)c2cc(OCc3cnccn3)ccc2n1Cc1ccc(Cl)cc1

nearest known ligand 0.86

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 19/20 0.86
ALOX5 P09917 8/20 0.72
CYP3A4 P08684 3/20 0.72
CYP2C9 P11712 3/20 0.72
PTGES2 Q9H7Z7 1/20 0.64
CYP2D6 P10635 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9173601 0.92 ALOX5AP (1.00) ALOX5APALOX5CYP3A4CYP2C9CYP2D6
SCHEMBL9305628 0.91 ALOX5AP (0.87) ALOX5APALOX5CYP3A4CYP2C9CYP2D6
SCHEMBL9178524 0.89 ALOX5AP (0.71) ALOX5APALOX5CYP3A4CYP2C9PTGES2
SCHEMBL9447569 0.89 ALOX5AP (0.87) ALOX5APALOX5CYP3A4CYP2C9CYP2D6
SCHEMBL9315369 0.85 ALOX5AP (0.86) ALOX5APALOX5CYP3A4CYP2C9PTGES2
SCHEMBL9044184 0.84 PTGES2 (0.78) ALOX5APALOX5CYP3A4CYP2C9PTGES2
SCHEMBL9185735 0.84 ALOX5AP (0.86) ALOX5APALOX5CYP3A4CYP2C9CYP2D6
SCHEMBL9305053 0.84 ALOX5AP (1.00) ALOX5APALOX5CYP3A4CYP2C9CYP2D6
SCHEMBL9387952 0.83 ALOX5AP (0.88) ALOX5APALOX5CYP3A4CYP2C9CYP2D6
SCHEMBL9388776 0.83 ALOX5AP (0.87) ALOX5APALOX5CYP3A4CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389650-A Antiinflammatory agents, anticoagulants, antispasmodic agents MERCK FROSST CANADA, INC. (CA) 1995-02-14 US disclosed
WO-1994013662-A1 (AZAARYLMETHOXY)INDOLES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-06-23 WO disclosed