SCHEMBL9181745

SCHEMBL9181745

OC(COc1ccnc2ccccc12)CN1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 4/20 0.64
KMT2A Q03164 7/20 0.63
MEN1 O00255 6/20 0.63
ALDH1A1 P00352 3/20 0.59
LMNA P02545 3/20 0.59
ALOX15 P16050 2/20 0.59
TSHR P16473 2/20 0.59
USP2 O75604 2/20 0.59
HTT P42858 2/20 0.59
TP53 P04637 1/20 0.59
GAA P10253 1/20 0.59
THRB P10828 1/20 0.59
MAPT P10636 3/20 0.56
ADRB2 P07550 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
KCNH2 Q12809 4/20 0.54
CYP2D6 P10635 1/20 0.53
NPSR1 Q6W5P4 1/20 0.52
OPRM1 P35372 1/20 0.51
OPRD1 P41143 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9183346 0.94 ABCB1 (0.74) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9183180 0.90 ABCB1 (0.69) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9184024 0.90 ABCB1 (0.69) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9187504 0.88 ABCB1 (0.67) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9186185 0.88 ABCB1 (0.67) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9183197 0.87 ABCB1 (0.68) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9186615 0.86 ABCB1 (0.64) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9183862 0.85 ABCB1 (0.63) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL9186444 0.85 ABCB1 (0.63) ABCB1KMT2AMEN1ALDH1A1LMNA
SCHEMBL14347213 0.85 ABCB1 (0.73) ABCB1KMT2AMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405843-A Anticancer drug potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1995-04-11 US disclosed
US-5204348-A Quinoline derivatives MITSUI TOATSU CHEMICALS INC. (JP) 1993-04-20 US disclosed
US-5112817-A Anticancer Drug Potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1992-05-12 US disclosed
EP-0363212-A2 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-04-11 EP disclosed