SCHEMBL9186129

SCHEMBL9186129

CC(C)(C)OC(=O)NC1C2CCN(C(=O)OCc3ccccc3)CC21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
PDE4B Q07343 1/20 0.50
HTT P42858 1/20 0.50
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HSD11B1 P28845 1/20 0.46
GRIN2B Q13224 2/20 0.45
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
GPR119 Q8TDV5 1/20 0.45
STS P08842 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
SYK P43405 1/20 0.44
CTSL P07711 1/20 0.44
MEN1 O00255 1/20 0.44
PARP1 P09874 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9186123 1.00 SMN1; SMN2 (0.51) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL28550674 0.95 SMN1; SMN2 (0.57) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL26077281 0.95 SMN1; SMN2 (0.57) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL28546986 0.95 SMN1; SMN2 (0.57) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL523499 0.92 PDE4B (0.54) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL523841 0.92 PDE4B (0.54) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL3547026 0.92 PDE4B (0.54) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL12527110 0.92 PDE4B (0.54) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL523500 0.92 PDE4B (0.54) SMN1; SMN2NPC1RAB9APDE4BHTT
SCHEMBL30965777 0.87 SMN1; SMN2 (0.49) SMN1; SMN2NPC1RAB9APDE4BHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0413455-B1 Azabicyclo quinolone carboxylic acids PFIZER (US) 1995-06-21 EP disclosed
US-5391763-A 3-aza-bicyclo[3.1.0]hexanes which are intermediates for anti-bacterial azabicyclo quinolone carboxylic acids PFIZER INC. (US) 1995-02-21 US disclosed
US-5229396-A Anti-bacterial azabicyclo quinolone carboxylic acids PFIZER INC. (US) 1993-07-20 US disclosed
EP-0413455-A2 Azabicyclo quinolone carboxylic acids PFIZER INC. (US) 1991-02-20 EP disclosed