SCHEMBL9186136

SCHEMBL9186136

CC(=O)N1CC(=O)NC(=Cc2ccc([N+](=O)[O-])cc2)C1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
MEN1 O00255 1/20 0.55
HRH3 Q9Y5N1 1/20 0.53
CASP3 P42574 1/20 0.44
METAP1 P53582 1/20 0.43
USP18 Q9UMW8 2/20 0.40
UCHL5 Q9Y5K5 2/20 0.40
AKR1B1 P15121 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KIF11 P52732 1/20 0.39
HSP90AA1 P07900 1/20 0.39
USP2 O75604 1/20 0.39
MAPT P10636 4/20 0.38
ALDH1A1 P00352 3/20 0.38
LMNA P02545 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
APP P05067 1/20 0.38
SNCA P37840 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9186135 1.00 KMT2A (0.55) KMT2AMEN1HRH3CASP3METAP1
SCHEMBL6132768 0.86 MEN1 (0.54) KMT2AMEN1HRH3METAP1HSP90AA1
SCHEMBL6132766 0.86 MEN1 (0.54) KMT2AMEN1HRH3METAP1HSP90AA1
SCHEMBL8596084 0.86 MEN1 (0.54) KMT2AMEN1HRH3METAP1HSP90AA1
SCHEMBL79547 0.82 MEN1 (0.66) KMT2AMEN1HRH3MAPTALDH1A1
SCHEMBL1598877 0.82 MEN1 (0.66) KMT2AMEN1HRH3MAPTALDH1A1
SCHEMBL7362683 0.82 MEN1 (0.66) KMT2AMEN1HRH3MAPTALDH1A1
SCHEMBL8592053 0.80 MEN1 (0.57) KMT2AMEN1HRH3METAP1TDP1
SCHEMBL8411263 0.80 HRH3 (0.64) KMT2AMEN1HRH3METAP1AKR1B1
SCHEMBL8411264 0.80 HRH3 (0.64) KMT2AMEN1HRH3METAP1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672036-A1 PHARMACEUTICALLY ACTIVE DIKETOPIPERAZINES XENOVA LIMITED (GB) 1995-09-20 EP disclosed
WO-1994004513-A1 PHARMACEUTICALLY ACTIVE DIKETOPIPERAZINES XENOVA LIMITED (GB) 1994-03-03 WO disclosed