Isosorbide Mononitrate

Isosorbide Mononitrate

SCHEMBL919022

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nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GUCY1A1GUCY1A2GUCY1B1GUCY1B2

The experimentally established mechanism targets of Isosorbide Mononitrate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.93
ALDH1A1 P00352 1/20 0.72
BCHE P06276 6/20 0.55
GSR P00390 7/20 0.48
CA2 P00918 1/20 0.47
THRB P10828 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isosorbide Mononitrate SCHEMBL8893344 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL5482432 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL616518 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL12238510 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL8894719 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL23906861 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL12787633 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL26782 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL22067709 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2
Isosorbide Mononitrate SCHEMBL8893635 0.96 MAPT (1.00) MAPTALDH1A1BCHEGSRCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11389534-B2 Methods of treating a subject for a condition PALO ALTO INVESTORS (US) 2022-07-19 US disclosed
US-10946197-B2 Treatment of conditions through modulation of the autonomic nervous system PALO ALTO INVESTORS (US) 2021-03-16 US disclosed
US-10702533-B2 Treatment of conditions through pharmacological modulation of the autonomic nervous system PALO ALTO INVESTORS (US) 2020-07-07 US disclosed
US-10086071-B2 Methods of treating a subject for a condition PALO ALTO INVESTORS (US) 2018-10-02 US disclosed
US-20170128457-A1 Treatment of Conditions Through Pharmacological Modulation of the Autonomic Nervous System PALO ALTO INVESTORS 2017-05-11 US disclosed
US-9585851-B2 Treatment of conditions through pharmacological modulation of the autonomic nervous system PALO ALTO INVESTORS (US) 2017-03-07 US disclosed
US-20160367807-A1 Treatment of Conditions Through Modulation of the Autonomic Nervous System PALO ALTO INVESTORS 2016-12-22 US disclosed
US-20140086872-A1 Methods of Treating a Subject for a Condition PALO ALTO INVESTORS (US) 2014-03-27 US disclosed
US-20120270876-A1 Treatment of Conditions Through Pharmacological Modulation of the Autonomic Nervous System PALO ALTO INVESTORS 2012-10-25 US disclosed
US-20110256097-A1 Treatment of Conditions that Increase in Severity and/or Occurrence During One or More Phases of the Menstrual Cycle PALO ALTO INVESTORS 2011-10-20 US disclosed
US-7899527-B2 Treatment of conditions through modulation of the autonomic nervous system during at least one predetermined menstrual cycle phase PALO ALTO INVESTORS (US) 2011-03-01 US disclosed
US-20110015188-A1 Treatment of Seasonal Conditions PALO ALTO INVENTORS 2011-01-20 US disclosed
US-20100286734-A1 Treatment of Conditions Through Modulation of the Autonomic Nervous System PALO ALTO INVESTORS 2010-11-11 US disclosed
US-20100260669-A1 Treatment of Seasonal Conditions Through Modulation of the Autonomic Nervous System PALO ALTO INVESTORS 2010-10-14 US disclosed
US-7738952-B2 Treatment of conditions through modulation of the autonomic nervous system PALO ALTO INVESTORS (US) 2010-06-15 US disclosed
US-20100119482-A1 Treatment of Conditions Through Modulation of the Autonomic Nervous System During at Least One Predetermined Menstrual Cycle Phase PALO ALTO INVESTORS 2010-05-13 US disclosed
US-20050256028-A1 Treatment of conditions through modulation of the autonomic nervous system during at least one predetermined menstrual cycle phase PALO ALTO INVESTORS 2005-11-17 US disclosed
US-20050240241-A1 Treatment of conditions through modulation of the autonomic nervous system PALO ALTO INVESTORS 2005-10-27 US disclosed
US-20050153885-A1 administering aldosterone antagonists such as spironolactone and eplerenone, to increasing the parasympathetic and sympathetic activity PALO ALTO INVESTORS 2005-07-14 US disclosed
US-20050143378-A1 Treatment of conditions through pharmacological modulation of the autonomic nervous system PALO ALTO INVESTORS 2005-06-30 US disclosed