SCHEMBL9190835

SCHEMBL9190835

N#Cc1ccc(C(CCO)c2ccc(F)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.59
CYP19A1 P11511 10/20 0.55
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
CYP2J2 P51589 1/20 0.49
CACNA1F O60840 2/20 0.44
HTR1A P08908 2/20 0.44
ADORA3 P0DMS8 2/20 0.44
DRD2 P14416 2/20 0.44
DRD1 P21728 2/20 0.44
DRD4 P21917 2/20 0.44
DRD5 P21918 2/20 0.44
HRH2 P25021 2/20 0.44
ADRA1D P25100 2/20 0.44
HTR2A P28223 2/20 0.44
HTR7 P34969 2/20 0.44
ADRA1A P35348 2/20 0.44
HRH1 P35367 2/20 0.44
ADRA1B P35368 2/20 0.44
OPRM1 P35372 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3637472 0.85 CYP19A1 (0.44) EPHX2CYP19A1CNR1
SCHEMBL6699187 0.80 CYP19A1 (0.49) CYP19A1HTR2AHRH1CACNA1C
SCHEMBL23126408 0.79 EPHX2 (0.51) EPHX2CYP19A1CYP2C9CYP2C19CYP2J2
SCHEMBL8411269 0.78 EPHX2 (0.58) EPHX2CYP19A1CYP2C9CYP2C19CYP2J2
SCHEMBL1349663 0.76 KDM4E (0.48) EPHX2CYP19A1CYP2C9CYP2C19CYP2J2
SCHEMBL5948050 0.75 EPHX2 (1.00) EPHX2CYP2C9CYP2C19CYP2J2
SCHEMBL13813062 0.75 CA12 (0.46) EPHX2CYP19A1MAOAMAOBKDM4E
SCHEMBL13891122 0.74 CA12 (0.41) EPHX2CYP19A1KDM4E
SCHEMBL12444126 0.74
SCHEMBL39936 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674626-A1 NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS ORION-YHTYMÄ OY (FI) 1995-10-04 EP disclosed