SCHEMBL9196751

SCHEMBL9196751

CCOC(=O)c1ccc(C=C(C)c2ccc3c(c2)SCCCS3)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 9/20 0.54
RARG P13631 9/20 0.54
RARA P10276 8/20 0.54
RXRA P19793 1/20 0.44
HPGD P15428 2/20 0.42
HTT P42858 2/20 0.42
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
LMNA P02545 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 1/20 0.40
MAOA P21397 1/20 0.40
PRKCA P17252 1/20 0.38
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9196746 1.00 RARB (0.54) RARBRARGRARARXRAHPGD
SCHEMBL9142983 0.95 RARB (0.56) RARBRARGRARARXRAHPGD
SCHEMBL9142979 0.95 RARB (0.56) RARBRARGRARARXRAHPGD
SCHEMBL9148441 0.88 RARB (0.52) RARBRARGRARARXRAHPGD
SCHEMBL9148433 0.88 RARB (0.52) RARBRARGRARARXRAHPGD
SCHEMBL9145537 0.87 RARG (0.48) RARBRARGRARARXRAHPGD
SCHEMBL9145541 0.87 RARG (0.48) RARBRARGRARARXRAHPGD
SCHEMBL9144382 0.87 RARB (0.51) RARBRARGRARARXRAHPGD
SCHEMBL9144389 0.87 RARB (0.51) RARBRARGRARARXRAHPGD
SCHEMBL9143264 0.86 RARB (0.53) RARBRARGRARARXRAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0350846-B1 Condensed heterocyclic compounds and their use in therapy HOFFMANN LA ROCHE (CH) 1995-10-11 EP claimed
US-5037825-A Useful In The Treatment Of Neoplasms, Dermatoses And Aging Of The Skin HOFFMANN-LA ROCHE INC. (US) 1991-08-06 US claimed