SCHEMBL9200539

SCHEMBL9200539

NCCN1C=Cc2ccccc2C1NCCNCCO

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.31
BRD4 O60885 1/20 0.31
CCL2 P13500 1/20 0.31
GRIN1 Q05586 3/20 0.30
GRIN2A Q12879 3/20 0.30
GRIN2B Q13224 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9198898 0.93 GRIN1 (0.34) HTR2AGRIN1GRIN2AGRIN2B
SCHEMBL28824445 0.67 BRD4 (0.40) HTR2ABRD4CCL2
SCHEMBL27951331 0.60 BRD4 (0.37) HTR2ASMN1; SMN2BRD4CCL2
SCHEMBL11155913 0.58 BRD4 (0.49) HTR2ASMN1; SMN2BRD4CCL2
Ethylenediamine SCHEMBL8371784 0.57 CA12 (0.53) SMN1; SMN2
SCHEMBL16078964 0.57 ACE2 (0.63)
Diethanolamine SCHEMBL1043915 0.57 SMN1; SMN2 (0.50) SMN1; SMN2
SCHEMBL10694747 0.56 BRD4 (0.55) HTR2ASMN1; SMN2BRD4CCL2
SCHEMBL7570833 0.56 BRD4 (0.42) HTR2ASMN1; SMN2BRD4CCL2
SCHEMBL10688105 0.56 BRD4 (0.46) HTR2ASMN1; SMN2BRD4CCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0662076-A1 2-AMINOALKYL-5-AMINOALKYLAMINO SUBSTITUTED ISOQUINOINDAZOLE-6-(2H)-ONES WITH ANTITUMOUR ACTIVITY THE UNIVERSITY OF VERMONT (US) 1995-07-12 EP claimed