SCHEMBL9204802

SCHEMBL9204802

C/C=C/Cc1cc(C/C=C/C)c(OC)c(/C=C/C(=O)c2ccc(N)cc2)c1O.CCOc1c(C)cc(C)c(O)c1/C=C/C(=O)c1ccc(N)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
KRAS P01116 1/20 0.43
KDM4E B2RXH2 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CYP1A1 P04798 3/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2D6 P10635 3/20 0.38
CYP1B1 Q16678 3/20 0.38
PTPN1 P18031 2/20 0.38
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9204807 1.00 CA1 (0.43) CA1CA2KRASKDM4ELMNA
SCHEMBL9203705 0.94 MAOB (0.42) KDM4ELMNAMAPTALDH1A1SMN1; SMN2
SCHEMBL9203700 0.94 MAOB (0.42) KDM4ELMNAMAPTALDH1A1SMN1; SMN2
SCHEMBL7183517 0.90 CA1 (0.42) CA1CA2KRASKDM4ELMNA
SCHEMBL7183516 0.90 CA1 (0.42) CA1CA2KRASKDM4ELMNA
SCHEMBL7188103 0.89 CA1 (0.52) CA1CA2KRASKDM4ELMNA
SCHEMBL7188097 0.89 CA1 (0.52) CA1CA2KRASKDM4ELMNA
SCHEMBL7185369 0.86 CA1 (0.46) CA1CA2KRASCTSLCTSB
SCHEMBL7185365 0.86 CA1 (0.46) CA1CA2KRASCTSLCTSB
SCHEMBL7191429 0.82 ABCG2 (0.49) KDM4ELMNAMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed