SCHEMBL9212178

SCHEMBL9212178

N#CN/C(=N\C(c1ccccc1)c1ccccc1)c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 1/20 0.47
EPHX2 P34913 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP2C19 P33261 2/20 0.42
CYP2C9 P11712 1/20 0.42
CYP3A4 P08684 1/20 0.41
POLB P06746 1/20 0.41
PLOD2 O00469 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HTT P42858 1/20 0.40
LMNA P02545 1/20 0.40
APP P05067 1/20 0.39
GAA P10253 1/20 0.39
HCAR3 P49019 1/20 0.39
HCAR2 Q8TDS4 1/20 0.39
CFTR P13569 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9212201 1.00 S1PR3 (0.47) S1PR3EPHX2KMT2ACYP2C19CYP2C9
Hydrochloric Acid SCHEMBL9211779 0.99 S1PR3 (0.46) S1PR3EPHX2KMT2ACYP2C19CYP2C9
Hydrochloric Acid SCHEMBL9211777 0.99 S1PR3 (0.46) S1PR3EPHX2KMT2ACYP2C19CYP2C9
SCHEMBL9208909 0.84 CYP2C9 (0.42) EPHX2KMT2ACYP2C19CYP2C9CYP3A4
SCHEMBL9213965 0.84 CYP2C9 (0.42) EPHX2KMT2ACYP2C19CYP2C9CYP3A4
Hydrochloric Acid SCHEMBL9217997 0.83 CYP2C9 (0.41) EPHX2KMT2ACYP2C19CYP2C9CYP3A4
Hydrochloric Acid SCHEMBL9218004 0.83 CYP2C9 (0.41) EPHX2KMT2ACYP2C19CYP2C9CYP3A4
SCHEMBL9211715 0.83 EPHX2 (0.46) EPHX2KMT2ACYP2C19CYP2C9CYP3A4
SCHEMBL9211713 0.83 EPHX2 (0.46) EPHX2KMT2ACYP2C19CYP2C9CYP3A4
Hydrochloric Acid SCHEMBL9218712 0.82 EPHX2 (0.45) EPHX2CYP2C19CYP2C9CYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP claimed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP claimed
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP disclosed
US-5272164-A Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1993-12-21 US disclosed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US disclosed
US-5166347-A Hypotensive agents, cardiovascular disorders, antiischemic agents and anticoagulants KIRIN BEER KABUSHIKI KAISHA (JP) 1992-11-24 US disclosed