SCHEMBL9213630

SCHEMBL9213630

COc1cc2c(cc1OC)CN(CC1CCCCN(CCc3ccc4ccccc4c3)C1)CC2

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 14/20 0.53
ABCG2 Q9UNQ0 6/20 0.53
DHCR7 Q9UBM7 2/20 0.49
HRH3 Q9Y5N1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214620 0.99 ABCB1 (0.52) ABCB1ABCG2DHCR7HRH3
Hydrochloric Acid SCHEMBL9215875 0.93 ABCB1 (0.54) ABCB1ABCG2DHCR7
SCHEMBL9204667 0.92 ABCB1 (0.48) ABCB1ABCG2DHCR7
SCHEMBL9207036 0.89 HRH3 (0.50) ABCB1ABCG2HRH3
Hydrochloric Acid SCHEMBL9214060 0.87 DHCR7 (0.48) ABCB1ABCG2DHCR7HRH3
SCHEMBL9211025 0.87 HRH3 (0.49) ABCB1ABCG2HRH3
SCHEMBL9215240 0.86 MEN1 (0.47) ABCB1HRH3
Hydrochloric Acid SCHEMBL9205960 0.86 DHCR7 (0.61) ABCB1ABCG2DHCR7
SCHEMBL9211431 0.85 HRH3 (0.47) ABCB1ABCG2HRH3
Hydrochloric Acid SCHEMBL9740420 0.85 CYP3A4 (0.47) ABCB1ABCG2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed