SCHEMBL9213709

SCHEMBL9213709

CCOC(=O)C(=CN(CC)CC)C(=O)c1cc(F)c(F)c(F)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.40
MEN1 O00255 4/20 0.40
NPSR1 Q6W5P4 4/20 0.40
LMNA P02545 4/20 0.40
MAPT P10636 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GAA P10253 2/20 0.35
DHODH Q02127 2/20 0.35
ALDH1A1 P00352 1/20 0.34
GLO1 Q04760 1/20 0.34
MAPK1 P28482 2/20 0.34
S1PR4 O95977 1/20 0.34
S1PR1 P21453 1/20 0.34
HTT P42858 1/20 0.34
STAT3 P40763 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9562231 1.00 KMT2A (0.40) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL10551891 0.94 KMT2A (0.37) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL30843044 0.88 MEN1 (0.40) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL4567521 0.88 MEN1 (0.40) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL3695378 0.88 MEN1 (0.40) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL9561731 0.88 MEN1 (0.40) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL17350379 0.88 KMT2A (0.36) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL17350817 0.86 KMT2A (0.41) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL12889528 0.85 MEN1 (0.44) KMT2AMEN1NPSR1LMNAMAPT
SCHEMBL10544905 0.82 NPSR1 (0.42) KMT2AMEN1NPSR1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0457090-B1 Process for the preparation of 3-amino-2 (het)aroyl-acrylic acid derivatives BAYER AG (DE) 1995-11-29 EP disclosed
US-5182401-A Bactericide intermediate BAYER AKTIENGESELLSCHAFT (DE) 1993-01-26 US disclosed
EP-0457090-A2 Process for the preparation of 3-amino-2 (het)aroyl-acrylic acid derivatives BAYER AG (DE) 1991-11-21 EP disclosed