SCHEMBL9218018

SCHEMBL9218018

Clc1ccc(N2CC=C(COc3ccc(C4=NCCO4)cc3)CC2)nn1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
LTA4H P09960 1/20 0.44
ACKR3 P25106 1/20 0.35
CYP1A2 P05177 1/20 0.33
BPTF Q12830 1/20 0.32
LSS P48449 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PANK3 Q9H999 1/20 0.31
KMT2A Q03164 1/20 0.31
AXL P30530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214015 0.78 HRH3 (0.65) KCNH2HRH3LTA4HACKR3
SCHEMBL9219081 0.73 KCNH2 (0.41) KCNH2HRH3KDM4EALDH1A1MAPT
SCHEMBL9219781 0.72 HRH3 (0.50) KCNH2HRH3LTA4HACKR3PANK3
SCHEMBL9211253 0.67 HRH3 (0.65) KCNH2HRH3LTA4HACKR3
SCHEMBL9211677 0.67 HRH3 (0.65) KCNH2HRH3LTA4HACKR3
SCHEMBL9216760 0.65 HRH3 (0.61) KCNH2HRH3LTA4HACKR3CYP1A2
SCHEMBL9311956 0.64 CYP1A2 (0.43) CYP1A2BPTFALDH1A1SMN1; SMN2KMT2A
SCHEMBL9213571 0.64 HRH3 (0.65) KCNH2HRH3LTA4HACKR3KDM4E
SCHEMBL9668080 0.63 HRH3 (0.68) KCNH2HRH3LTA4HACKR3KDM4E
SCHEMBL9217275 0.63 HRH3 (0.65) KCNH2HRH3LTA4HACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320032-B1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA NV (BE) 1995-01-18 EP disclosed
US-5231184-A Viricide intermediate JANSSEN PHARMACEUTICA N.V. (BE) 1993-07-27 US disclosed
US-5106973-A Viricide intermediates JANSSEN PHARMACEUTICA N.V. (BE) 1992-04-21 US disclosed
US-4992433-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-12 US disclosed