SCHEMBL9228261

SCHEMBL9228261

Nc1nc(N)c2c(n1)NC(CCCc1ccc(C(=O)N[C@@H](CCC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O)cc1)C2

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GART P22102 7/20 0.57
DHFR P00374 5/20 0.55
ATIC P31939 2/20 0.51
FOLR2 P14207 2/20 0.49
FOLR1 P15328 2/20 0.49
SLC46A1 Q96NT5 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844865 0.97 GART (0.60) GARTDHFRATIC
SCHEMBL9229346 0.95 GART (0.54) GARTDHFRATIC
SCHEMBL9219257 0.93 GART (0.57) GARTDHFRATICFOLR2FOLR1
SCHEMBL9844758 0.92 GART (0.57) GARTDHFRATIC
SCHEMBL9844788 0.90 GART (0.60) GARTDHFRATICFOLR2FOLR1
SCHEMBL9223490 0.88 GART (0.54) GARTDHFRATIC
SCHEMBL9228277 0.87 GART (0.51) GARTDHFRATIC
SCHEMBL9844755 0.84 GART (0.57) GARTDHFRATIC
SCHEMBL9446047 0.84 GART (0.69) GARTDHFRATIC
SCHEMBL9229354 0.82 GART (0.48) GARTDHFRATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5459129-A Antitumor agents; enzyme inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-17 US disclosed
US-5268362-A Containing benzene and purine rings TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-07 US disclosed
EP-0492316-A1 Condensed heterocyclic oligoglutamate derivatives, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1992-07-01 EP disclosed