SCHEMBL9237136

SCHEMBL9237136

N[C@H](C(=O)O)C(CC(=O)O)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.51
GAA P10253 1/20 0.51
CYP2C9 P11712 1/20 0.51
PKM P14618 1/20 0.51
CYP2C19 P33261 1/20 0.51
PPARG P37231 12/20 0.50
PPARA Q07869 10/20 0.50
MAPT P10636 1/20 0.43
SLC1A5 Q15758 1/20 0.42
SLC1A3 P43003 1/20 0.42
SLC1A2 P43004 1/20 0.42
SLC1A1 P43005 1/20 0.42
MMP12 P39900 2/20 0.42
MMP13 P45452 1/20 0.42
FFAR1 O14842 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9237130 1.00 CYP1A2 (0.51) CYP1A2GAACYP2C9PKMCYP2C19
SCHEMBL9241640 0.91 KMT2A (0.44) CYP1A2CYP2C9CYP2C19PPARGPPARA
SCHEMBL9241636 0.91 KMT2A (0.44) CYP1A2CYP2C9CYP2C19PPARGPPARA
SCHEMBL9233763 0.88 FFAR1 (0.45) FFAR1
SCHEMBL9233755 0.88 FFAR1 (0.45) FFAR1
SCHEMBL9238843 0.88 PPARG (0.50) PPARGPPARAMMP12MMP13FFAR1
SCHEMBL9238852 0.88 PPARG (0.50) PPARGPPARAMMP12MMP13FFAR1
SCHEMBL9238489 0.85 PPARG (0.55) CYP1A2CYP2C9CYP2C19PPARGPPARA
SCHEMBL9237967 0.85 PPARG (0.55) CYP1A2CYP2C9CYP2C19PPARGPPARA
SCHEMBL9237973 0.85 PPARG (0.55) CYP1A2CYP2C9CYP2C19PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1108240-A Excitatory amino acid receptor antagonists LILLY CO ELI (US) 1995-09-13 CN disclosed
EP-0658539-A1 Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 1995-06-21 EP disclosed