SCHEMBL9237307

SCHEMBL9237307

Cc1ccc(-c2ccc(NC(=O)OC(C)(C)C)cn2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.48
PTPN1 P18031 5/20 0.48
PTPN2 P17706 2/20 0.47
PSMB8 P28062 1/20 0.46
NAMPT P43490 1/20 0.46
PTPN6 P29350 1/20 0.46
PTPN11 Q06124 1/20 0.46
MAP4K4 O95819 1/20 0.46
BCL2 P10415 2/20 0.44
SREBF2 Q12772 1/20 0.43
AURKA O14965 1/20 0.43
ABL1 P00519 1/20 0.43
NTRK1 P04629 1/20 0.43
LCK P06239 1/20 0.43
CSF1R P07333 1/20 0.43
RET P07949 1/20 0.43
MET P08581 1/20 0.43
PDGFRB P09619 1/20 0.43
PIM1 P11309 1/20 0.43
PDGFRA P16234 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5776405 0.88 PTPN1 (0.55) CYP17A1PTPN1PTPN2PSMB8NAMPT
SCHEMBL9235573 0.85 CYP17A1 (0.53) CYP17A1PTPN1PTPN2PSMB8NAMPT
SCHEMBL16492878 0.82 CYP17A1 (0.50) CYP17A1PTPN1SREBF2
SCHEMBL178373 0.81 CYP17A1 (0.54) CYP17A1PSMB8NAMPTCA12CA1
SCHEMBL38655104 0.81 CYP17A1 (0.52) CYP17A1PTPN1PTPN2PSMB8NAMPT
SCHEMBL29153845 0.80 BCL2 (0.42) CYP17A1PTPN1PTPN2PSMB8NAMPT
SCHEMBL28103663 0.80 TDP1 (0.59) PTPN1PTPN2PTPN6PTPN11AURKA
SCHEMBL30208803 0.80 NAMPT (0.56) CYP17A1PSMB8NAMPTMAP4K4MAPKAPK2
SCHEMBL376258 0.80 NAMPT (0.56) CYP17A1PSMB8NAMPTMAP4K4MAPKAPK2
SCHEMBL12582106 0.79 PTPN2 (0.48) CYP17A1PTPN1PTPN2NAMPTMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665223-A1 Antitumor agent, novel 3(2H)-pyridazinone derivatives and their preparation TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-02 EP disclosed