SCHEMBL9246765

SCHEMBL9246765

CCOC(=O)C(N)C1c2ccccc2Sc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.47
GAA P10253 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
PIN1 Q13526 1/20 0.39
TSHR P16473 4/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HSD17B10 Q99714 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
NOX1 Q9Y5S8 1/20 0.37
CACNA1C Q13936 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
MMP8 P22894 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9244137 0.99 BCHE (0.46) BCHEGAAMEN1KMT2ANPC1
SCHEMBL25301977 0.83 CYP1A2 (0.44) MEN1KMT2ANPC1PIN1TSHR
SCHEMBL30522607 0.83 CYP1A2 (0.44) MEN1KMT2ANPC1PIN1TSHR
SCHEMBL9243385 0.81 TACR1 (0.45) GAAMEN1KMT2ANPC1PIN1
SCHEMBL9545140 0.79 POLB (0.51) MEN1KMT2ANPC1TSHRKDM4E
SCHEMBL18816035 0.79 TACR1 (0.46) MEN1KMT2ANPC1PIN1TSHR
Hydrochloric Acid SCHEMBL9241964 0.78 TACR1 (0.45) MEN1KMT2APIN1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL9241189 0.78 POLB (0.50) MEN1KMT2ANPC1TSHRKDM4E
SCHEMBL9246204 0.78 BCHE (0.43) BCHEGAAMEN1KMT2ANPC1
SCHEMBL9241143 0.78 GRM1 (0.42) BCHETSHRACHECYP1A2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5449778-A Peptide intermediates WARNER-LAMBERT COMPANY (US) 1995-09-12 US disclosed
EP-0637305-A1 NOVEL CYCLIC AMINO ACIDS AND DERIVATIVES THEREOF WARNER-LAMBERT COMPANY (US) 1995-02-08 EP disclosed
US-5264577-A Cyclic amino acids and derivatives thereof WARNER-LAMBERT COMPANY (US) 1993-11-23 US disclosed
WO-1993021176-A1 NOVEL CYCLIC AMINO ACIDS AND DERIVATIVES THEREOF WARNER-LAMBERT COMPANY (US) 1993-10-28 WO disclosed