SCHEMBL9254840

SCHEMBL9254840

CCCC/C=C/[C@H]1CC[C@H](CC[C@H]2CC[C@H](c3ccc(F)c(F)c3)CC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SGPL1 O95470 3/20 0.36
S1PR1 P21453 2/20 0.36
CYP2C9 P11712 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
SLC10A2 Q12908 1/20 0.32
HCRTR2 O43614 3/20 0.31
CCR2 P41597 1/20 0.31
ESR2 Q92731 1/20 0.31
KDM1A O60341 1/20 0.31
SPHK1 Q9NYA1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254847 1.00 SGPL1 (0.36) SGPL1S1PR1CYP2C9ALDH1A1LMNA
SCHEMBL9311979 0.93 CYP2C9 (0.36) SGPL1S1PR1CYP2C9ALDH1A1LMNA
SCHEMBL8518689 0.93 CYP2C9 (0.36) SGPL1S1PR1CYP2C9ALDH1A1LMNA
SCHEMBL8518687 0.93 CYP2C9 (0.36) SGPL1S1PR1CYP2C9ALDH1A1LMNA
SCHEMBL8518684 0.93 CYP2C9 (0.36) SGPL1S1PR1CYP2C9ALDH1A1LMNA
SCHEMBL9254740 0.93 CYP2C9 (0.36) SGPL1S1PR1CYP2C9ALDH1A1LMNA
SCHEMBL9481226 0.90 SGPL1 (0.36) SGPL1S1PR1SLC10A2HCRTR2KDM1A
SCHEMBL9481233 0.90 SGPL1 (0.36) SGPL1S1PR1SLC10A2HCRTR2KDM1A
SCHEMBL9319900 0.90 SGPL1 (0.36) SGPL1S1PR1SLC10A2HCRTR2KDM1A
SCHEMBL9319888 0.90 SGPL1 (0.36) SGPL1S1PR1SLC10A2HCRTR2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5454974-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1995-10-03 US disclosed
US-5302317-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1994-04-12 US disclosed
EP-0315014-B1 Halogenated benzene derivatives HOFFMANN LA ROCHE (CH) 1994-01-12 EP disclosed
EP-0315050-B1 ALCENYL BICYCLOHEXANES F. HOFFMANN-LA ROCHE AG (CH) 1993-09-01 EP disclosed
US-5230826-A HALOBENZENE LIQUID CRYSTALS HOFFMANN-LA ROCHE INC. (US) 1993-07-27 US disclosed
US-5013477-A Alkenylbicyclohexane liquid crystals HOFFMANN-LA ROCHE INC. (US) 1991-05-07 US disclosed