SCHEMBL9258940

SCHEMBL9258940

c1cc(-c2n[nH]c3ccncc23)ccn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.57
PIM1 P11309 3/20 0.54
LRRK2 Q5S007 4/20 0.51
IDO1 P14902 2/20 0.51
NTRK1 P04629 1/20 0.49
JAK2 O60674 1/20 0.47
CLK2 P49760 3/20 0.47
DYRK1A Q13627 3/20 0.47
CLK3 P49761 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
ALPL P05186 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
TTK P33981 1/20 0.47
MAPK10 P53779 1/20 0.47
MAPK1 P28482 3/20 0.47
MAP2K4 P45985 1/20 0.46
MAPK3 P27361 2/20 0.46
PIM3 Q86V86 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1513103 0.89 IDO1 (0.63) MKNK1PIM1LRRK2IDO1CLK2
SCHEMBL1921806 0.85 MKNK1 (0.47) MKNK1PIM1LRRK2IDO1CLK2
SCHEMBL9251358 0.85 CLK2 (0.54) MKNK1PIM1LRRK2IDO1JAK2
SCHEMBL1922328 0.85 MAP2K4 (0.56) MKNK1PIM1LRRK2IDO1CLK2
SCHEMBL1922154 0.85 MAPK14 (0.51) MKNK1LRRK2IDO1NTRK1CLK2
Hydrochloric Acid SCHEMBL9260992 0.84 MKNK1 (0.46) MKNK1PIM1LRRK2IDO1CLK2
SCHEMBL2242478 0.81 LRRK2 (0.59) MKNK1LRRK2IDO1
SCHEMBL10533662 0.80 IDO1 (0.74) MKNK1PIM1LRRK2IDO1NTRK1
SCHEMBL27817994 0.79 MAPT (0.59) MKNK1PIM1LRRK2IDO1ALDH1A1
SCHEMBL15543826 0.78 PIM1 (0.52) MKNK1PIM1LRRK2IDO1CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428169-A Antidepressants, treating compulsive disorders, stuttering, trichotillomania HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-06-27 US disclosed
US-5380847-A Reaction of 1-methylpiperidine-4-hydrazine, ketone and titanium isopropoxide to form hydrazone HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1995-01-10 US disclosed
EP-0594001-A1 Pyrazolo 4,3-c pyridines, a process for their preparation and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-04-27 EP disclosed
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US disclosed
US-5264576-A Antiserotonin agents, antidepressants and obsessive-compulsive disorders HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-11-23 US disclosed