SCHEMBL9267697

SCHEMBL9267697

CC(=O)c1ccc2c(c1)C(Cc1ccncc1)(Cc1ccncc1)c1ccccc1-2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 5/20 0.57
CYP3A4 P08684 3/20 0.57
ALOX15 P16050 2/20 0.57
TSHR P16473 2/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2C9 P11712 2/20 0.57
PDK2 Q15119 8/20 0.51
S100A4 P26447 1/20 0.42
ATM Q13315 1/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
KCNH2 Q12809 1/20 0.41
ALDH1A1 P00352 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
THPO P40225 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9266879 0.99 KCNQ2 (0.56) KCNQ2CYP3A4ALOX15TSHRCYP1A2
Hydrochloric Acid SCHEMBL9261182 0.83 PDK2 (0.54) KCNQ2CYP3A4ALOX15TSHRCYP1A2
SCHEMBL18012748 0.80 PDK2 (0.58) PDK2S100A4NPC1MAPTRAB9A
SCHEMBL9261740 0.80 KCNQ2 (0.79) KCNQ2CYP3A4ALOX15TSHRCYP1A2
SCHEMBL9266386 0.79 KCNQ2 (0.60) KCNQ2CYP3A4ALOX15TSHRCYP1A2
Hydrochloric Acid SCHEMBL9273003 0.78 KCNQ2 (0.59) KCNQ2CYP3A4ALOX15TSHRCYP1A2
SCHEMBL17084359 0.78 PDK2 (0.56) PDK2S100A4NPC1MAPTRAB9A
SCHEMBL9264288 0.78 KCNQ2 (0.59) KCNQ2CYP3A4ALOX15TSHRCYP1A2
Hydrochloric Acid SCHEMBL9265822 0.78 KCNQ2 (0.77) KCNQ2CYP3A4ALOX15TSHRCYP1A2
SCHEMBL9269302 0.76 KCNQ2 (0.54) KCNQ2CYP3A4ALOX15TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311010-B1 Alpha,Alpha-disubstituted aromatics and heteroaromatics as cognition enhancers DU PONT MERCK PHARMA (US) 1994-02-02 EP claimed
US-5434264-A α,α-disubstituted aromatics and heteroaromatics as cognition enhancers THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-07-18 US disclosed
US-5300642-A α, α-disubstituted aromatics and heteroaromatics as cognition enhancers THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-04-05 US disclosed
EP-0311010-B1 Alpha,Alpha-disubstituted aromatics and heteroaromatics as cognition enhancers DU PONT MERCK PHARMA (US) 1994-02-02 EP disclosed
EP-0532054-A1 Process for preparing alpha,alpha-disubstituted aromatics and heteroaromatics as cognition enhancers THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-03-17 EP disclosed
US-5173489-A α,α-disubstituted aromatics and heteroaromatics as cognition enhancers THE DUPONT MERCK PHARMACEUTICAL CO. (US) 1992-12-22 US disclosed
EP-0311010-A2 Alpha,Alpha-disubstituted aromatics and heteroaromatics as cognition enhancers THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1989-04-12 EP disclosed