SCHEMBL9268672

SCHEMBL9268672

CCCC(=O)/C(=C/Nc1ccccc1COC(=O)c1ccc(OC)cc1)C(=O)OCC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.47
DHODH Q02127 1/20 0.47
LMNA P02545 4/20 0.46
MAPT P10636 3/20 0.46
KDM4E B2RXH2 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
ALDH1A1 P00352 6/20 0.45
HPGD P15428 3/20 0.45
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 1/20 0.43
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9268678 1.00 GAA (0.47) GAADHODHLMNAMAPTKDM4E
SCHEMBL9264530 0.91 GAA (0.52) GAADHODHLMNAMAPTKDM4E
SCHEMBL9264524 0.91 GAA (0.52) GAADHODHLMNAMAPTKDM4E
SCHEMBL10532873 0.81 PPARG (0.42) GAADHODHLMNAMAPTCYP3A4
SCHEMBL9268172 0.80 DHODH (0.59) GAADHODHLMNAMAPTKDM4E
SCHEMBL9268176 0.80 DHODH (0.59) GAADHODHLMNAMAPTKDM4E
SCHEMBL9270355 0.80 GAA (0.47) GAADHODHLMNAMAPTKDM4E
SCHEMBL10533835 0.78 DHODH (0.56) GAADHODHLMNAMAPTKDM4E
SCHEMBL9723914 0.78 DHODH (0.59) GAADHODHLMNAMAPTKDM4E
SCHEMBL9652064 0.78 NPSR1 (0.63) GAADHODHLMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5432182-A Inhibitors of gastric acid secretion SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-07-11 US disclosed
EP-0330485-B1 4-AMINO-3-ACYL QUINOLINE DERIVATIVES AND THEIR USE AS INHIBITORS OF GASTRIC ACID SECRETION SmithKline Beecham Intercredit B.V. (NL) 1993-05-26 EP disclosed
US-5089504-A SUBSTITUTED 4-AMINOQUINOLINE DERIVATIVES AS GASTRIC ACID SECRETION INHIBITORS SMITHKLINE BECKMAN INTERCREDIT B.V. (NL) 1992-02-18 US disclosed
EP-0330485-A1 4-Amino-3-acyl quinoline derivatives and their use as inhibitors of gastric acid secretion SmithKline Beecham Intercredit B.V. (NL) 1989-08-30 EP disclosed