Tandutinib

Tandutinib

SCHEMBL927974

COc1cc2c(N3CCN(C(=O)Nc4ccc(OC(C)C)cc4)CC3)ncnc2cc1OCCCN1CCCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FLT3KITPDGFRB

The experimentally established mechanism targets of Tandutinib. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB known ✓ P09619 19/20 1.00
FLT3 known ✓ P36888 7/20 1.00
KIT known ✓ P10721 6/20 1.00
CSF1R P07333 4/20 1.00
PLK4 O00444 1/20 1.00
GAK O14976 1/20 1.00
EPHB6 O15197 1/20 1.00
STK10 O94804 1/20 1.00
EGFR P00533 1/20 1.00
NTRK1 P04629 1/20 1.00
LCK P06239 1/20 1.00
FGFR1 P11362 1/20 1.00
SRC P12931 1/20 1.00
PDGFRA P16234 1/20 1.00
FLT1 P17948 1/20 1.00
FGFR2 P21802 1/20 1.00
FGFR4 P22455 1/20 1.00
FGFR3 P22607 1/20 1.00
AXL P30530 1/20 1.00
FLT4 P35916 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tandutinib SCHEMBL29393910 1.00 PDGFRB (1.00) PDGFRBFLT3KITCSF1RPLK4
Tandutinib SCHEMBL2478362 0.99 PDGFRB (0.98) PDGFRBFLT3KITCSF1RPLK4
SCHEMBL13330466 0.99 PDGFRB (1.00) PDGFRBFLT3KITCSF1RPLK4
Tandutinib SCHEMBL2496722 0.96 PDGFRB (0.93) PDGFRBFLT3KITCSF1RPLK4
SCHEMBL13330462 0.96 PDGFRB (1.00) PDGFRBFLT3KITCSF1RPLK4
SCHEMBL13524739 0.94 PDGFRB (0.90) PDGFRBFLT3KITCSF1RPLK4
SCHEMBL13529590 0.93 PDGFRB (0.89) PDGFRBFLT3KITCSF1RPLK4
SCHEMBL13330482 0.93 PDGFRB (0.88) PDGFRBFLT3KITCSF1RPLK4
SCHEMBL29460355 0.93 PDGFRB (1.00) PDGFRBFLT3KITCSF1RPLK4
SCHEMBL317630 0.93 PDGFRB (1.00) PDGFRBFLT3KITCSF1RPLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2602 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260142007-A1 DIGITAL THERAPEUTICS AND COMBINATION THERAPY FOR THE TREATMENT OF TENOSYNOVIAL GIANT CELL TUMOR (TGCT) REMEPY HEALTH LTD (IL) 2026-05-21 US claimed
EP-4743086-A2 TREATING MYELOID DISORDERS Mayo Foundation for Medical Education and Research (US) 2026-05-20 EP claimed
EP-4731220-A2 METHODS OF TREATING CHRONIC LYMPHOCYTIC LEUKEMIA Dana Farber Cancer Institute, Inc. (US) 2026-04-29 EP claimed
EP-4719387-A2 COMPLEMENT ANTIBODY-DRUG CONJUGATES ADS Therapeutics LLC (US) 2026-04-08 EP claimed
EP-4722388-A1 PREDICTION OF AN OUTCOME OF A SUBJECT SUFFERING FROM ACUTE MYOLOID LEUKEMIA Koninklijke Philips N.V. (NL) 2026-04-08 EP claimed
US-20250333795-A1 COMPOSITION FOR AMPLIFYING FLT3 GENE, AND USES THEREOF NGENEBIO (KR) 2025-10-30 US claimed
US-20250281624-A1 METHODS AND COMPOSITIONS FOR TREATING CHRONIC INFLAMMATORY INJURY, METAPLASIA, DYSPLASIA AND CANCERS OF EPITHELIAL TISSUES UNIVERSITY OF HOUSTON SYSTEM (US) 2025-09-11 US claimed
US-20250213497-A1 A NANO IN MICRO FORMULATION AND PROCESS THEREOF AMRITA VISHWA VIDYAPEETHAM (IN) 2025-07-03 US claimed
EP-4578962-A1 COMPOSITION FOR AMPLIFYING FLT3 GENE, AND USES THEREOF Ngenebio (KR) 2025-07-02 EP claimed
WO-2025131038-A1 COMPOSITIONS AND METHODS FOR DELIVERY OF PHARMACEUTICAL ACTIVES ADS THERAPEUTICS LLC (US) 2025-06-26 WO claimed
EP-2638896-A1 Cationic liposomal drug delivery system for specific targeting of human cd14+ monocytes in whole blood Bioneer A/S (DK) 2013-09-18 EP claimed
US-20110293615-A1 Use of Combination of Anti-Angiogenic Substance and c-kit Kinase Inhibitor EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-12-01 US claimed
US-20090053236-A1 USE OF COMBINATION OF ANTI-ANGIOGENIC SUBSTANCE AND c-kit KINASE INHIBITOR EISAI R & D MANAGEMENT CO., LTD. (JP) 2009-02-26 US claimed
EP-1949902-A1 USE OF COMBINATION OF ANTI-ANGIOGENIC SUBSTANCE AND c-kit KINASE INHIBITOR Eisai R&D Management Co., Ltd. (JP) 2008-07-30 EP claimed
JP-2005533604-A 2005-11-10 JP claimed
US-20050203612-A1 Luminal prostheses which allow for programmed and controlled delivery of mycophenolic acid or derivatives with increased efficacy to selected locations within a patient's vasculature to inhibit restenosis and hyperplasia AVANTEC VASCULAR CORPORATION (US) 2005-09-15 US claimed
EP-1539041-A1 DEVICES DELIVERING THERAPEUTIC AGENTS AND METHODS REGARDING THE SAME Avantec Vascular Corporation (US) 2005-06-15 EP claimed
WO-2005051229-A2 DEVICES DELIVERING THERAPEUTIC AGENTS AND METHODS REGARDING THE SAME AVANTEC VASCULAR CORPORATION (US) 2005-06-09 WO claimed
US-20050125054-A1 Devices delivering therapeutic agents and methods regarding the same AVANTEC VASCULAR CORPORATION (US) 2005-06-09 US claimed
WO-2004010900-A1 DEVICES DELIVERING THERAPEUTIC AGENTS AND METHODS REGARDING THE SAME AVANTEC VASCULAR CORPORATION (US) 2004-02-05 WO claimed