SCHEMBL9280955

SCHEMBL9280955

COc1ccc(CN2C(=O)NC(C#Cc3ccccn3)(C3CC3)c3cc(Cl)ccc32)cc1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.42
PTGDR2 Q9Y5Y4 5/20 0.40
EDNRB P24530 3/20 0.37
EDNRA P25101 3/20 0.37
ALDH1A1 P00352 2/20 0.37
ADAMTS5 Q9UNA0 2/20 0.36
OPRL1 P41146 1/20 0.36
MMP12 P39900 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALOX15 P16050 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9542846 0.85 PTGDR2 (0.43) SCN9APTGDR2ALDH1A1ADAMTS5OPRL1
SCHEMBL9571243 0.83 PTGDR2 (0.42) SCN9APTGDR2EDNRBEDNRAALDH1A1
SCHEMBL9571197 0.82 PTGDR2 (0.43) SCN9APTGDR2ALDH1A1OPRL1KDM4E
SCHEMBL9144120 0.81 PTGDR2 (0.46) SCN9APTGDR2ALDH1A1OPRL1KDM4E
SCHEMBL9571203 0.80 PTGDR2 (0.46) SCN9APTGDR2EDNRBEDNRAALDH1A1
SCHEMBL9541552 0.76 PTGDR2 (0.49) SCN9APTGDR2ALDH1A1OPRL1KDM4E
SCHEMBL9571205 0.75 PTGDR2 (0.38) SCN9APTGDR2EDNRBEDNRAALDH1A1
SCHEMBL9541586 0.75 PTGDR2 (0.45) SCN9APTGDR2EDNRBEDNRAOPRL1
SCHEMBL9542788 0.74 PTGDR2 (0.47) SCN9APTGDR2EDNRBEDNRAALDH1A1
SCHEMBL9539775 0.74 PTGDR2 (0.44) SCN9APTGDR2ALDH1A1OPRL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5457201-A Chiral resolution process MERCK & CO., INC. (US) 1995-10-10 US disclosed
EP-0569083-A1 New quinazolines as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-11-10 EP disclosed