SCHEMBL9290245

SCHEMBL9290245

Cc1cc(Cl)cc(C(=O)NC(C)C)c1NC(=O)C1CC(C(F)(F)F)=NN1c1ncccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 10/20 0.40
RBP4 P02753 1/20 0.35
TRPV1 Q8NER1 3/20 0.34
CSF1R P07333 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9289364 0.94 MALT1 (0.36) MALT1RBP4TRPV1CSF1R
SCHEMBL13003161 0.92 MALT1 (0.37) MALT1RBP4TRPV1
SCHEMBL12295362 0.92 MALT1 (0.37) MALT1RBP4TRPV1
SCHEMBL13356332 0.92 MALT1 (0.37) MALT1RBP4TRPV1CSF1R
SCHEMBL9290237 0.91 MALT1 (0.41) MALT1RBP4TRPV1
SCHEMBL9289044 0.91 MALT1 (0.36) MALT1RBP4TRPV1CSF1R
SCHEMBL9289370 0.91 MALT1 (0.39) MALT1RBP4TRPV1CSF1R
SCHEMBL9289365 0.90 MALT1 (0.42) MALT1
SCHEMBL13338276 0.90 MALT1 (0.42) MALT1RBP4TRPV1
SCHEMBL9290071 0.89 MALT1 (0.42) MALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197844-B1 SPIROHETEROCYCLIC PYRROLIDINE DIONE DERIVATIVES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-07-25 EP disclosed
WO-2012092827-A1 CHEMICAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2012-07-12 WO disclosed
WO-2012069008-A1 3-SUBSTITUTED SPIROHETEROCYCLIC FURAN AND THIOFURAN DIONE DERIVATIVES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-31 WO disclosed
WO-2011113756-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2011-09-22 WO disclosed
WO-2011095462-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2011-08-11 WO disclosed
EP-2332411-A1 Fungicidal compositions Syngenta Participations AG (CH) 2011-06-15 EP disclosed
WO-2011067203-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067135-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067131-A1 SPIROHETEROCYCLIC DIONE DERIVATIVES USED AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
EP-2213167-A1 Anthranilamide derivatives and their use for the control of insects and acari Syngenta Participations AG (CH) 2010-08-04 EP disclosed
WO-2010066780-A1 SPIROHETEROCYCLIC N-OXYPIPERIDINES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-17 WO disclosed
WO-2010063670-A1 SPIROHETEROCYCLIC N-OXYAMIDES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-10 WO disclosed
EP-2099785-B1 N-CYANOALKYLANTHRANILAMIDES AS INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-05-19 EP disclosed
EP-1984354-B1 PESTICIDES CONTAINING A BICYCLIC BISAMIDE STRUCTURE SYNGENTA PARTICIPATIONS AG (CH) 2009-08-05 EP disclosed
WO-2009049851-A1 SPIROHETEROCYCLIC PYRROLIDINE DIONE DERIVATIVES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-04-23 WO disclosed
WO-2009024341-A2 CONDENSED ANTHRAN I LAMI DE DERIVATIVES AS INSECTISIDES SYNGENTA PARTICIPATIONS AG, (CH) 2009-02-26 WO disclosed
WO-2009021717-A2 PESTICIDAL FORMULATION SYNGENTA PARTICIPATIONS AG (CH) 2009-02-19 WO disclosed
WO-2009010260-A2 CONDENSED ANTHRANILAMIDE INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-01-22 WO disclosed
WO-2008064891-A1 N-CYANOALKYLANTHRANILAMIDES AS INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2008-06-05 WO disclosed