SCHEMBL9301346

SCHEMBL9301346

S=C=Nc1cccc(OCc2ccc3ccccc3n2)c1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYSLTR1 Q9Y271 10/20 0.60
GPBAR1 Q8TDU6 7/20 0.60
CYSLTR2 Q9NS75 4/20 0.60
PDE10A Q9Y233 1/20 0.59
TP53 P04637 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
MAPK1 P28482 1/20 0.52
CYP2C19 P33261 1/20 0.52
HIF1A Q16665 1/20 0.52
ALOX5 P09917 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10512475 0.79 PDE10A (0.77) CYSLTR1GPBAR1CYSLTR2PDE10ACYP1A2
SCHEMBL6088376 0.77 CYSLTR1 (0.72) CYSLTR1GPBAR1CYSLTR2PDE10A
SCHEMBL10547998 0.76 CYSLTR1 (1.00) CYSLTR1GPBAR1CYSLTR2PDE10A
SCHEMBL6744402 0.76 CYSLTR1 (0.69) CYSLTR1GPBAR1CYSLTR2PDE10ATP53
SCHEMBL10545363 0.76 CYSLTR1 (0.71) CYSLTR1GPBAR1CYSLTR2PDE10ATP53
SCHEMBL9047808 0.76 CYSLTR1 (0.69) CYSLTR1GPBAR1CYSLTR2PDE10ACYP1A2
SCHEMBL10690028 0.76 CYSLTR1 (0.69) CYSLTR1GPBAR1CYSLTR2PDE10ATP53
Hydrogen Sulfide SCHEMBL9818428 0.76 CYSLTR1 (0.71) CYSLTR1GPBAR1CYSLTR2PDE10A
SCHEMBL10510977 0.76 CYSLTR1 (0.69) CYSLTR1GPBAR1CYSLTR2PDE10ATP53
SCHEMBL10513942 0.76 CYSLTR1 (0.69) CYSLTR1GPBAR1CYSLTR2PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360909-A THROMBOXANE A2 ANTAGONIST TERUMO KABUSHIKI KAISHA (JP) 1994-11-01 US disclosed
EP-0562796-A1 Phenoxyacetic acid compounds and medical preparations containing them TERUMO KABUSHIKI KAISHA (JP) 1993-09-29 EP disclosed